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4-[(4,6-dimethylquinolin-2-yl)amino]butan-1-ol
2-[4-(3,6-dimethylpyrazin-2-yl)-1H-pyrazol-1-yl]-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
2-(3-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
methyl 1-{3-[(4-ethoxyphenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
1-[(4-fluorophenyl)methyl]-N-[3-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
3-{[1-(4,4,4-trifluorobutanoyl)pyrrolidin-3-yl]methyl}benzoic acid
2-(3-chloro-4-hydroxyphenyl)-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(3S,4S)-N-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-methoxypyrrolidin-3-amine
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-(6-methylpyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(cyclopropylmethyl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
N-benzyl-N,1-dimethyl-5-[methyl(1,2-oxazol-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-(2-phenoxyethyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
6-methyl-5-{5-[3-(trifluoromethyl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
3-(2,6-dimethylphenyl)-1-{[1-(oxan-4-yl)piperidin-3-yl]methyl}urea
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-2-phenylacetamide
3-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(2-hydroxyethyl)amino)-1λ6-thiolane-1,1-dione
N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]pyridazine-4-carboxamide
2-[(3-methoxyphenyl)methyl]-4-[4-(1H-pyrazol-3-yl)benzoyl]morpholine
N-(2,3-dihydro-1H-inden-2-yl)-3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanamide
3-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-1-(2-methoxyethyl)-1-(pyridin-4-ylmethyl)urea
N3-[3-(4-fluorophenyl)propyl]piperidine-1,3-dicarboxamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(2-oxopyrrolidin-1-yl)acetamide
N-(1-carbamoylcycloheptyl)-4-propylpyrimidine-5-carboxamide
methyl 4-[(4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]benzoate
4-({3-[6-(thiomorpholin-4-yl)pyridazin-3-yl]phenyl}methyl)morpholine
2-fluoro-N-[1-(pyrazin-2-yl)propan-2-yl]-5-sulfamoylbenzamide
9-[2-(dimethylamino)propanoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3R,4S)-1-[(2-chlorophenyl)methanesulfonyl]-4-cyclopropylpyrrolidin-3-yl]acetamide
1-methyl-4-(1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)piperazine
[(3-{[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(thiophen-3-ylmethyl)amine
4-(4-methylphenyl)-N-[1-(pyrazin-2-yl)propan-2-yl]-5-(pyridin-4-yl)pyrimidin-2-amine
1-(azepan-1-yl)-3-{4-[(4-fluoropiperidin-1-yl)methyl]-2-methoxyphenoxy}propan-2-ol
N3-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-N5-cyclohexyl-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]-3-methoxy-2,2-dimethylpropan-1-one
2-(2,3-dimethoxyphenyl)-2-{[2-(1H-imidazol-1-yl)ethyl](methyl)amino}acetic acid
(1H-imidazol-2-ylmethyl)(methyl){[5-(2-phenylethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
8-[4-(4-chlorophenyl)butanoyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
methyl 6-cyclohexanecarbonyl-2-[(3-fluoro-4-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(1S,3R)-3-cyclopropanesulfonamido-N-[(dimethyl-1,2-oxazol-4-yl)methyl]cyclopentane-1-carboxamide
6-ethyl-3-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-1,5-dimethyl-1,2-dihydropyridin-2-one
N-methyl-5-{[2-(1H-pyrazol-1-yl)butanamido]methyl}-1,2,4-oxadiazole-3-carboxamide
N-{1-[1-(oxan-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
2-[5-(4-cyanooxan-4-yl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
2-(2-aminoacetyl)-N-methyl-N-(pyridin-3-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
4-{2-[(4-fluorophenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
3-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-(2-fluoro-5-methylphenyl)-3-methylurea
3-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)-1-(propan-2-yl)piperidine-4-carboxamide
5-methanesulfonyl-1'-(pyridine-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]