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1-(2,3-dimethylquinoxalin-6-yl)-3-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}urea
5-(1-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}pyrrolidin-2-yl)-3-methyl-1H-1,2,4-triazole
6-{[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}quinoline
N-({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
8-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1-benzyl-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(1-carbamoylethyl)-1-(3-methylbutyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
2-methyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1,3-thiazole-4-carboxamide
N-[(1S)-2-(1H-imidazol-4-yl)-1-[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]ethyl]acetamide
(3aR,7aS)-2-[6-(4-fluorophenyl)pyridazin-3-yl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-methylpropan-1-one
3-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-6-methyl-1,2-dihydropyridin-2-one
N-(2-{[3-(3-hydroxy-3-methylbutyl)phenyl]formamido}ethyl)acetamide
1-cyclopentyl-4-[4-(4-methylthiophen-2-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
(1S,4S)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-propyl-5-{[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]methyl}pyrimidin-2-amine
4-[(2E)-2-methylbut-2-en-1-yl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3aR,5R,6S,7aS)-2-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}-octahydro-1H-isoindole-5,6-diol
1-[(5-methylfuran-2-yl)methyl]-4-oxo-N3-(prop-2-en-1-yl)-N5-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
9-(cyclopropylmethyl)-1-methyl-10-oxo-N-phenyl-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
1-{[(3R,4R)-4-(hydroxymethyl)-1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]pyrrolidin-3-yl]methyl}piperidin-4-ol
1-(2-chloroprop-2-en-1-yl)-6,7-dimethoxy-3-[({[2-(trifluoromethyl)phenyl]methyl}amino)methyl]-1,2-dihydroquinolin-2-one
8-[3-(3-hydroxy-3-methylbutyl)benzoyl]-2-methyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-(3-ethylphenyl)-4-(4-methylpiperidin-1-yl)-4-oxobutanamide
4-hydroxy-N-[(3-methyl-1-benzofuran-2-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
3-methyl-6-[5-(3-propyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]pyridazine
2-(2-hydroxyethyl)-9-[1-oxo-1-(pyrrolidin-1-yl)propan-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
2-(4-phenylphenyl)-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}ethan-1-one
1-(2-fluoro-4-methylbenzoyl)-3-(3-methoxypropyl)piperidine
N-[2-(1,3-benzothiazol-2-yl)ethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
3-{2-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-{3-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-oxopropyl}-3,4-dihydroquinazolin-4-one
3-[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]-N-(4-methylphenyl)-3-oxopropanamide
2-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
8-{2-amino-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-methyl-1-{3-[2-(morpholine-4-carbonyl)piperazin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
(5S,9aS,9bS)-5-[5-(methoxymethyl)furan-2-yl]-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-ethyl-6-(4-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperazin-1-yl)pyridine-3-carboxamide
2-[4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-1-yl]pyrazine
8-(1-benzofuran-2-ylmethyl)-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperazin-1-yl]-1,3-benzothiazole
(3S,4S)-4-methyl-1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidine-3,4-diol
2-[4-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
4-[4-(4-cyclopentyl-1,4-diazepane-1-carbonyl)phenyl]-2-methylbutan-2-ol
4-[(2S)-2-amino-2-[3-methyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]ethyl]phenol
1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
[(1-{[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]urea
ethyl 1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-4-(2-methoxyethyl)piperidine-4-carboxylate
{1-[({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}(methyl)amino)methyl]cyclobutyl}methanol