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2-{4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
2-[4-(pentan-3-yl)piperazin-1-yl]-N-(prop-2-en-1-yl)pyridine-3-carboxamide
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
(3R,4R)-1-(1-benzofuran-2-ylmethyl)-4-(4-methylpiperazin-1-yl)piperidin-3-ol
5-{[2-(3-hydroxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
{[2-methoxy-5-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenyl]methyl}(methyl)amine
5-fluoro-2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-N,N-dimethylpyrimidin-4-amine
(2R,6R)-10-methoxy-4-[3-(1H-pyrazol-1-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
4-methyl-3-[4-(1H-pyrazol-5-yl)phenyl]pyridine
2-(morpholin-3-yl)-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide
5-{6-amino-5-cyano-4-[3-(methoxycarbonyl)-1H-pyrazol-4-yl]pyridin-2-yl}thiophene-3-carboxylic acid
1-[1-(2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]propan-1-ol
4-({4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyridine
(2R,6R)-4-[(dimethyl-1,3-thiazol-5-yl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(4-{[4-(2-methylphenyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)(pyridin-3-yl)methanol
[5-(1,3-benzoxazol-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methanamine
{[2-(methoxymethyl)pyrimidin-5-yl]methyl}(3-phenylprop-2-yn-1-yl)propylamine
N-[4-(1H-indol-3-yl)butan-2-yl]-1-methanesulfonylpiperidin-4-amine
2-ethyl-8-[2-(2,2,2-trifluoro-1-phenylethoxy)acetyl]-2,8-diazaspiro[4.5]decan-3-one
(2S,4S)-4-amino-N-methyl-1-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]pyrrolidine-2-carboxamide
(2R)-2-phenyl-2-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}ethan-1-ol
2-(4-{[2-(furan-2-yl)phenyl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
7-(cyclobutylmethyl)-2-[4-(1H-imidazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-methyl-3-(1H-pyrazol-1-yl)propanamide
(4aS,8aS)-2-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
2-(2-methoxyethyl)-8-(3-methoxypropanoyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
2,6-dimethyl-N-[1-(1H-pyrazol-1-yl)propan-2-yl]quinoline-3-carboxamide
N,4-dimethyl-5-[3-(2-methylphenoxymethyl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
2-oxo-8-(pyridine-4-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-(1-ethyl-1H-imidazol-2-yl)-1-[4-(pyrrolidin-1-ylmethyl)benzoyl]piperidine
4-ethyl-1-{2-[3-(trifluoromethyl)phenyl]acetyl}-1,4-diazepan-5-one
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
3-acetamido-N-[2-(2-ethoxyethoxy)phenyl]pyrrolidine-1-carboxamide
N-{[8-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(2,3-dimethylphenyl)methyl]piperidine-3-carboxamide
methyl 7-oxo-9-[2-(thiophen-2-yl)ethoxy]-3-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-cyclohexyl-4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-(furan-2-ylmethyl)-2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetamide
4-(3-acetylbenzoyl)-5-methyl-1-(3-methylphenyl)piperazin-2-one
2-[(2-hydroxyethyl)({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})amino]ethan-1-ol
(2R,3R)-3-(2,5-dihydro-1H-pyrrol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
1-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)but-3-en-1-one
N-methyl-4-oxo-1-(3-phenylpropyl)-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridine-3-carboxamide
[(4-methanesulfonylphenyl)methyl](methyl)[(5-phenyl-1,2-oxazol-3-yl)methyl]amine
5-fluoro-2-{1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-2-yl}-1H-1,3-benzodiazole
3-(2-fluorophenyl)-5-(furan-3-ylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
4-[4-(furan-2-carbonyl)-1,4-diazepane-1-carbonyl]-1-oxaspiro[4.5]decan-2-one