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3-(4-hydroxyphenyl)-N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-1H-pyrazole-5-carboxamide
methyl(pyridin-3-ylmethyl){[5-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}amine
2-(3-cyclopropanecarbonyl-1H-indol-1-yl)-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]acetamide
N,N-dimethyl-2-[(1S,5R)-6-[(1-propyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
1-(3-ethyl-1H-pyrazole-4-carbonyl)-3-(3-methoxypropyl)piperidine
1-cyclopropyl-N-methyl-6-oxo-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-3-carboxamide
4-(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperazin-2-one
3-cyclohexyl-1-(7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
2-({2-[1-(thiophene-2-sulfonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(dimethylamino)-N-[3-(3-methyl-1H-pyrazol-1-yl)propyl]-2-(3-methylphenyl)acetamide
3-{2-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]propyl}pyridine
(2E)-3-(1-methyl-1H-pyrazol-4-yl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}prop-2-en-1-one
(1S,5R)-6-[(1-methyl-1H-indol-6-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-methoxy-2-{[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}phenol
4-(3-fluorophenoxy)-1-(thiophene-2-carbonyl)piperidine-4-carboxylic acid
methyl[(4-methyl-1H-imidazol-2-yl)methyl]{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
N-cyclohexyl-N-methyl-4-(4-propylpiperazin-1-yl)pyridine-2-carboxamide
2-(4-methyl-1H-pyrazol-1-yl)-1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]ethan-1-one
1-[6-(2-methoxyphenyl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
2-(dimethyl-1,3-thiazol-5-yl)-N-{[3-(trifluoromethoxy)phenyl]methyl}acetamide
N-[(2R,4R,6S)-2-(4-chlorophenyl)-6-[2-(methylamino)pyridin-3-yl]oxan-4-yl]acetamide
N-(2-ethylphenyl)-4-[5-(4-methoxybenzamido)-1H-pyrazol-1-yl]piperidine-1-carboxamide
N-(2-methoxyethyl)-N,1-dimethyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[(2R)-2-aminopropanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(2S,4R)-4-{[(3,4-difluorophenyl)methyl]amino}-N-ethyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
1-{4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
2-(1H-imidazol-2-yl)-1-(2-methoxy-5-methylphenyl)-1H-imidazole
2-(cyclopropylmethyl)-9-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-2-(pyridin-3-yl)morpholine
(3R,4R)-1-(4-cyclopentylpyrimidin-2-yl)-3,4-dimethylpyrrolidin-3-ol
N-[(3-methylphenyl)methyl]-N-(propan-2-yl)pyrrolidine-3-carboxamide
8-pentanoyl-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
6-[3-(3-ethylphenoxy)azetidin-1-yl]pyrimidin-4-amine
5-(4-methylphenyl)-N-[(1-methylpyrrolidin-3-yl)methyl]furan-2-carboxamide
N-(butan-2-yl)-N-[(4-chlorophenyl)methyl]propanamide
3-[5-({methyl[1-(3-phenylpropyl)piperidin-3-yl]amino}methyl)thiophen-2-yl]prop-2-yn-1-ol
2-methyl-4-{4-[3-(morpholin-4-yl)azetidine-1-carbonyl]phenyl}butan-2-ol
N-(2-methylbutan-2-yl)-5-{1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-{2-oxo-2-[3-(thiophene-2-carbonyl)piperidin-1-yl]ethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
5-{methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
methyl 2-[9-oxo-8-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carboxylate
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(1-phenylcyclopropanecarbonyl)-decahydro-1,6-naphthyridin-2-one
7-amino-4-(2,3-dimethyl-1H-indol-7-yl)-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
9-(2-hydroxyethyl)-1-methyl-4-[4-(trifluoromethyl)pyridin-2-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}dimethylamine
2-(3-hydroxypropyl)-9-(quinoxalin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
(1R,7S)-3-[(3-methylphenyl)methyl]-6-(5-oxo-1,4-diazepane-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-1H-indole
1-{4-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-1-carboxamide