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3-({4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
(2R,3R,6R)-5-cyclobutanecarbonyl-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{1-[(5-methylfuran-2-yl)methyl]-4-(1,2-oxazol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
N-{[7-(4-chlorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
(1R,5R)-6-benzyl-3-(6-methylpyridazin-3-yl)-3,6-diazabicyclo[3.2.2]nonane
[3-({[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)-2,4,6-trimethylphenyl]methyl acetate
5-[({[3-(2-{4-[3-(4-fluorophenyl)benzoyl]piperazin-1-yl}ethoxy)phenyl]methyl}(methyl)amino)methyl]pyrrolidin-2-one
4-(2-butoxybenzoyl)-1-(3-methoxyphenyl)piperazin-2-one
2-amino-N,4-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,3-thiazole-5-carboxamide
8-[(3-chloropyridin-4-yl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane
(1R,5R)-N,N-dimethyl-6-(1,2,3,4-tetrahydroquinoline-6-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-ethyl-2,3-dimethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
(3R,4R)-1-(4-chloro-2-methylbenzoyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
(3S,4S)-4-cyclopropyl-1-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]pyrrolidine-3-carboxylic acid
(2S,4R)-4-amino-1-[3-(benzylsulfanyl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
7-{[(2S)-2,4,5,5-tetramethylpiperazin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
5-(4-fluorophenyl)-3-[4-(2-phenoxyethyl)piperazin-1-yl]-1,2,4-triazine
N-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-2-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)acetamide
{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(quinoxalin-6-ylmethyl)amine
1-(pyrrolidin-1-yl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}cyclopentane-1-carboxamide
1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-3-(furan-2-yl)propan-1-one
2-{1-[(1R,7S)-3-[(3-methoxyphenyl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-6-yl]-N-methylformamido}-N-methylacetamide
4-ethyl-1-methyl-3-[1-(quinolin-2-yl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-[1-methyl-6-(propan-2-yloxy)-1H-indazol-3-yl]acetamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperazine
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]amino}methyl)piperidin-2-one
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[(3,5-dimethoxyphenyl)methyl]piperidine
3-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-{3-[(trifluoromethyl)sulfanyl]phenyl}urea
1-(carbamoylmethyl)-N-(cyclohex-1-en-1-ylmethyl)piperidine-3-carboxamide
2-({1-[(4-ethynylphenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
N,6-dimethyl-N-(2-methylpropyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
N-[(1-benzylpiperidin-3-yl)methyl]-1-(4-chlorophenyl)cyclopropane-1-carboxamide
2-ethoxy-4-({3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)phenol
[(2-ethoxy-5-{[(2S,5R)-5-(morpholin-4-ylmethyl)oxolan-2-yl]methyl}phenyl)methyl](methyl)amine
5-(4-methyl-1,4-diazepan-1-yl)-2-[2-(2-methyl-2,3-dihydro-1H-indol-1-yl)-2-oxoethyl]-2,3-dihydropyridazin-3-one
{1-[(5-chlorothiophen-2-yl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
5-[1-(cyclohexylmethyl)-4-hydroxypiperidin-4-yl]-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(3-methylpyrazin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-cyclopropyl-4-methyl-N-{[3-(oxolan-2-ylmethoxy)phenyl]methyl}benzamide
1-[3-(2-methylphenoxy)azetidin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
7-(2-methoxyacetamido)-1-methyl-2-phenyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
4,4,4-trifluoro-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylbutanamide
methyl 3-(2-methylpropyl)-2-oxo-1-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methylacetamide
1-(adamantan-2-yl)-4-[(2S,4S)-1-[(4-methoxy-3-methylphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]piperazine
2-propyl-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyridine-4-carboxamide
2-ethyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-(propan-2-yl)piperidine-4-carboxamide
N-(1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N,2-dimethylfuran-3-carboxamide