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1-(3-methylbut-2-en-1-yl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
(2E)-3-(4-methoxyphenyl)-N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)prop-2-enamide
1-(1-{6-[2-(dimethylamino)phenyl]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
[2-(1-methylpyrrolidin-2-yl)ethyl]({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl})amine
1-methyl-4-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
6-oxo-1-(pyridin-2-ylmethyl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]piperidine-3-carboxamide
2-{4-[(6-methoxy-2H-chromen-3-yl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
3-[2-(3-methoxyphenyl)ethyl]-1-(prop-2-ene-1-sulfonyl)piperidine
N6-cyclopentyl-N5-methyl-N5-[3-(morpholin-4-yl)propyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-({1-[(5-chlorofuran-2-yl)methyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
methyl 3-[(cyclohexylformamido)methyl]-5-(2-methoxyacetamido)benzoate
3-({[2-(dimethylamino)ethyl][(5-methylthiophen-2-yl)methyl]carbamoyl}amino)-4-methylbenzamide
5-({[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amino}methyl)-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(2-methoxyethyl)piperazin-1-yl]ethan-1-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-5-ethyl-2-methylpyrimidin-4-amine
N-methyl-2-(piperidin-1-yl)-N-(pyridin-2-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
5-[4-(4-acetylphenyl)piperazine-1-carbonyl]-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
methyl 1-(naphthalen-2-ylmethoxy)-2-oxo-8-(quinolin-4-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-cyclopentyl-N-methyl-N-(2-methylpropyl)-4-oxo-5-(3-oxo-4-phenylpiperazine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-2-amine
1-[2-methoxy-5-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
2-({[(3R,4R)-1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
3-[(propan-2-yl)sulfamoyl]-5-(quinolin-8-yl)benzoic acid
1-(diethylamino)-3-(2-methoxy-5-{[(1-phenylcyclopropyl)amino]methyl}phenoxy)propan-2-ol
3-[(3R,4S)-4-(dimethylamino)-1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-3-yl]propan-1-ol
6-{[benzyl(2-hydroxyethyl)amino]methyl}-N-[1-(naphthalen-1-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
4-methyl-1-(3-phenylpropyl)-1,4-diazepan-5-one
1-[(4-methoxyphenyl)methyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{[4-(pyridin-4-yl)phenyl]sulfanyl}acetamide
2-({2-[(3,4-dimethoxyphenyl)methyl]-1,3-benzoxazol-6-yl}formamido)acetamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-propyl-1,5-diazatricyclo[5.2.2.02,6]undecane
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl){[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}amine
6-(3-methylpyrazin-2-yl)-2-[3-(1,4-oxazepan-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
3-(6-methoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-N-(thiophen-2-ylmethyl)propanamide
1-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(methylamino)ethan-1-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]piperazine
4-[5-(1H-imidazol-4-ylmethyl)-3-phenyl-1H-1,2,4-triazol-1-yl]-3-methylpyridine
N4-[(1-methanesulfonylpiperidin-3-yl)methyl]-N2,N2-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
3-methyl-4-[1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidin-2-yl]-1,2,5-oxadiazole
1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-(1-methylpiperidin-4-yl)piperidine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[3-(3-hydroxypiperidin-1-yl)propyl]benzamide
5-(morpholin-4-ylmethyl)-N,N-bis(propan-2-yl)-1,2-oxazole-3-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
2-amino-4-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-7-methyl-5H,7H-furo[3,4-b]pyridine-3-carbonitrile
1-[(1,4-dimethyl-1H-pyrazol-5-yl)methyl]-N,N-diethylpiperidine-3-carboxamide
[4-(3-phenyl-1,2-oxazole-5-carbonyl)-1,4-oxazepan-6-yl]methanol
4-(2-chlorophenyl)-6-methylpyrimidin-2-amine
4-{1,5-dibenzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine