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N-ethyl-5-[(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)methyl]pyrimidin-2-amine
2-(hydroxymethyl)-N-methyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-1H-1,3-benzodiazole-5-carboxamide
(3S)-4-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)sulfonyl]-3-ethylmorpholine
3-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carbonyl]-1-methyl-1,4-dihydroquinolin-4-one
1-[2-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)ethyl]piperidine-3-carboxamide
2-(4-acetyl-1,4-diazepan-1-yl)-2-(2,3-dihydro-1-benzofuran-7-yl)acetic acid
8-(4-ethyl-5-methylpyrimidin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
1-benzyl-8-[3-(5-methylfuran-2-yl)butyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4R)-4-(4-fluorophenyl)-1-(3-propyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxylic acid
4-[(1E)-3-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}prop-1-en-1-yl]-2-methoxyphenol
N-[(1-methylpyrrolidin-3-yl)methyl]-6-(propan-2-yl)-1H-indole-2-carboxamide
1-(3-methoxybenzoyl)-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazine
methyl (2S)-3-methyl-2-{[(1-methylpiperidin-4-yl)(pyridin-4-ylmethyl)carbamoyl]amino}butanoate
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1-(propan-2-yl)piperidine-4-carboxamide
8-(2,1,3-benzothiadiazol-5-ylmethyl)-1-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1,3-dimethyl-6-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(dimethylamino)-N,4-dimethyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidine-5-carboxamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(3-fluorophenyl)-1,3-benzoxazole-5-carboxamide
N-[2-phenyl-2-(piperidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
N-(oxan-2-ylmethyl)-3-(pyridin-3-yl)propanamide
3-[(2-oxo-5,5-diphenylpiperidin-1-yl)methyl]-1λ6-thiolane-1,1-dione
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-3-(pyrrolidine-1-carbonyl)pyridin-2-amine
[(4-methanesulfonylphenyl)methyl](2-methoxyethyl)(thiophen-2-ylmethyl)amine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(2S)-oxolan-2-ylmethyl]propanamide
3-{5-[(1-propyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-(3-methoxyphenyl)-3-{1-[(1-methyl-1H-indol-3-yl)methyl]piperidin-4-yl}propanamide
ethyl 1-(3-methoxybenzoyl)-4-(2-phenylethyl)piperidine-4-carboxylate
methyl 6-{[(2-methoxyethyl)(methyl)amino]methyl}-3-[2-(3-methylphenyl)acetamido]thieno[2,3-b]pyridine-2-carboxylate
N-(1-{7-[(5-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
1-[7-(6,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-[(4-chlorophenyl)methyl]-4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-1,2,3-triazole
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
benzyl N-[1-(2-propyl-1,3-thiazole-4-carbonyl)pyrrolidin-3-yl]carbamate
2-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}pyridin-3-ol
1-{[2-(3-chlorophenyl)-6,7-dimethoxyquinolin-3-yl]methyl}piperidin-4-ol
1-(2-methylprop-2-en-1-yl)-5-oxopyrrolidine-3-carboxylic acid
1-[(3-methyl-1-benzofuran-2-yl)methyl]-4-(pyridin-3-ylmethyl)piperazine
1-[(1S,2R)-2-butylcyclopropanecarbonyl]-4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidine
N,N-diethyl-1-(3,5,7-trimethyl-1H-indole-2-carbonyl)pyrrolidin-3-amine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
[1-(1,3-thiazole-4-carbonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}urea
1-(2-chloro-5-fluorophenyl)-3-[1-(methoxymethyl)cyclopropyl]-3-methylurea
5-benzyl-N-(pyrrolidin-3-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-[5-(trifluoromethyl)pyridin-2-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
{[4-(difluoromethoxy)phenyl]methyl}({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
2-[4-(2,2-dimethylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-1-phenoxypropan-2-ol
N-(4-chloro-2-fluorophenyl)-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane-4-carboxamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide