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5-fluoro-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-(pyrrolidin-1-yl)pyrimidine
2-[3-cyclopropyl-5-(1-phenyl-1H-1,2,3-triazol-5-yl)-1H-1,2,4-triazol-1-yl]pyridine
1-cyclohexyl-4-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepane
2-(1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}piperidin-3-yl)-4-methyl-1H-1,3-benzodiazole
4-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]-1,2-dihydroisoquinolin-1-one
4-(4-fluorophenoxy)-1-(thiophene-2-carbonyl)piperidine
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-(4-methylpyridin-2-yl)piperazine
1-[2-chloro-5-(morpholine-4-carbonyl)phenyl]-3-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-methyl-3-phenylbutan-1-one
2-{5-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl}ethan-1-ol
5,6,7-trimethoxy-N,N-dimethyl-3-{[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]methyl}quinolin-2-amine
(2,1,3-benzothiadiazol-5-ylmethyl)[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amine
2-amino-1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-methylpropan-1-one
2-methyl-4-[4-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)phenyl]butan-2-ol
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-1-methyl-1H-pyrazole-3-carboxamide
{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
1-(1-{6-[4-(hydroxymethyl)phenyl]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one
3-benzyl-4-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
1-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-3-(1H-1,2,4-triazol-3-yl)urea
N-[(3S,4R)-1-[(5-acetylthiophen-3-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide
2,6-dimethoxy-N-[(3-methyloxetan-3-yl)methyl]pyridine-3-carboxamide
3-{3-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidin-1-yl]-3-oxopropyl}-5-methyl-2,3-dihydro-1,3-benzoxazol-2-one
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
3-(1H-indol-3-yl)-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)propanamide
4-[4-(oxan-4-yl)piperazine-1-carbonyl]benzene-1-sulfonamide
6-(4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperazin-1-yl)pyridine-3-carbonitrile
6-[2-chloro-3-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
3-(2-amino-1,3-thiazol-4-yl)-N-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}propanamide
methyl 1-(2-methoxyethoxy)-8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
3-[3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanoyl]-3,9-diazaspiro[5.6]dodecan-10-one
2-(dimethylamino)-2-(4-fluorophenyl)-1-[3-(3-methoxyphenoxy)azetidin-1-yl]ethan-1-one
5-{2-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]-2-oxoethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(1H-imidazol-2-ylmethyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine
3-{2-[4-(4-hydroxybut-1-yn-1-yl)phenyl]-1H-imidazol-1-yl}-N-methylbenzamide
N,N-dimethyl-3-[(6-oxo-1,6-dihydropyridin-3-yl)methyl]pyrrolidine-1-sulfonamide
4-[5-(methanesulfonylmethyl)pyridin-2-yl]aniline
2-{9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}-6-(propan-2-yl)pyridine-3-carbonitrile
7-[(4,5-dichlorothiophen-2-yl)sulfonyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(3aR,5S,6S,7aS)-2-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}-octahydro-1H-isoindole-5,6-diol
4-(2,5-di-tert-butylphenyl)-4H-1,2,4-triazole
5-cyclopropanecarbonyl-1'-(3,6-dimethylpyrazin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-cyclobutyl-2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carboxamide
5-fluoro-N4,N4-dimethyl-N2-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]pyrimidine-2,4-diamine
(3R,4R)-4-amino-1-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]piperidin-3-ol
N-[(2-fluorophenyl)methyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-{2-[5-(3-methylthiophen-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,2,3,4-tetrazole
3-[(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]pyridine
4-[(3-fluorophenyl)methyl]-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1,3-dimethyl-6-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(methoxymethyl)-N-[2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)ethyl]cyclobutane-1-carboxamide