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N,N-diethyl-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
5-chloro-N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
N-benzyl-N-(3-hydroxy-2-methylpropyl)-2-(methylamino)benzamide
N-benzyl-N-methyl-2-(pyrrolidine-1-carbonyl)-2,3-dihydro-1H-inden-2-amine
3-fluoro-4-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzene-1-sulfonamide
2-amino-4-cyclopropyl-6-(3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
11-[(1,3-benzothiazol-2-ylmethyl)amino]-4-[(4-fluorophenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-(oxan-4-yl)-N-[3-(2-oxopyrrolidin-1-yl)phenyl]piperazine-1-carboxamide
1'-(3-methoxypyrazin-2-yl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N,N-dimethyl-2-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
1-(3-{[3-(2-hydroxyethyl)-4-[1-(propan-2-yl)piperidin-4-yl]piperazin-1-yl]methyl}phenyl)ethan-1-one
1-(3,5-dimethylphenyl)-4-[2-hydroxy-2-(4-methoxyphenyl)acetyl]piperazin-2-one
(4aS,7aR)-1-(naphthalen-2-ylmethyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-N-[1-(thiophen-2-yl)ethyl]pyrimidin-2-amine
methyl 4-{[4-(2-methylphenyl)phenyl]carbamoyl}piperazine-1-carboxylate
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,1-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-N-(pyridin-3-ylmethyl)thiophene-2-carboxamide
N-({5-[3-(5-methylfuran-2-yl)butyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
N-({5-[(2-phenyl-1,3-thiazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
N-[(2-chlorophenyl)methyl]-2-ethyl-N-(propan-2-yl)pyrimidine-5-carboxamide
1-(2-ethoxyethyl)-5-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-3-methyl-1H-pyrazole
3-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
methyl (2R,4S)-1-[2-(benzyloxy)ethyl]-4-hydroxypiperidine-2-carboxylate
1-[2,5-difluoro-4-(trifluoromethyl)phenyl]-3-methyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]urea
2-(4-benzyl-3-butyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-methylacetamide
3-(5-benzyl-1,3,4-thiadiazol-2-yl)-1-[(4-fluorophenyl)methyl]-1-methylurea
(3S)-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-ol
methyl 4-[4-(3-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]benzoate
7-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-(hydroxymethyl)-1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperidin-4-ol
(2S)-1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-4-methyl-2-phenylpiperazine
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]piperidine
4-{[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidin-1-yl]methyl}-N-(1,3-thiazol-2-yl)benzamide
(3S,4S)-4-methoxy-N-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1-(propan-2-yl)pyrrolidin-3-amine
N-(1H-imidazol-2-ylmethyl)-N-methyl-1-(propan-2-yl)piperidine-4-carboxamide
3-{1-[2-(4-methanesulfonylphenyl)acetyl]piperidin-3-yl}benzoic acid
5,6-dimethyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)pyridine-3-carboxamide
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-2-(thiophen-2-yl)acetamide
1-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
6-(1-benzofuran-2-ylmethyl)-N-[2-(1H-imidazol-1-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}piperidin-3-yl)-1H-1,3-benzodiazole
5-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}pyrimidin-2-amine
N-[2-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-2-carboxamide
N-methyl-N-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-(hydroxymethyl)-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-ol
1-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-3-(1,3-dimethyl-4-phenyl-1H-pyrazol-5-yl)-1-methylurea
4-[1-(4-methyl-1H-imidazole-2-carbonyl)piperidin-4-yl]pyrimidin-2-amine
N-{2-[3-(3-methylbutyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]propyl}ethane-1-sulfonamide
3-methoxy-2-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridine