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[(2S,4R)-4-(dimethylamino)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]pyrrolidin-2-yl]methanol
3-(dimethylsulfamoyl)-N-[3-(1H-imidazol-1-yl)propyl]-5-[(quinolin-8-ylmethyl)amino]benzamide
1-(1-benzylpiperidin-4-yl)-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
2-{[3-(3-methoxyphenyl)-1H-pyrazol-5-yl]formamido}-3-phenylpropanoic acid
({4-cyclopropyl-5-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-[(3R,4S)-4-cyclopropyl-1-[3-(methylsulfanyl)propyl]pyrrolidin-3-yl]-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
2-(butylsulfanyl)-N4-[(5-methyl-1H-pyrazol-3-yl)methyl]pyrimidine-4,6-diamine
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-[4-(3-methylphenyl)piperazin-1-yl]acetamide
N-[(3R,4S)-4-(propan-2-yl)-1-[3-(4H-1,2,4-triazol-4-yl)propanoyl]pyrrolidin-3-yl]methanesulfonamide
3-{3-[1-(oxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine
3-[(3R,4S)-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]propanamide
1-ethyl-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-3,5-dimethyl-1H-pyrazole
2-[3-(2-methoxyethyl)-5-(4-propylpyrimidin-5-yl)-1H-1,2,4-triazol-1-yl]acetic acid
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
N-[2-(1H-indol-1-yl)ethyl]-N,3-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
methyl 3-[2-(2-phenylethyl)morpholine-4-carbonyl]benzoate
N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-5,6,7,8-tetrahydroquinoline-3-carboxamide
methyl 3-(2-methoxyacetamido)-5-({[3-(trifluoromethyl)phenyl]formamido}methyl)benzoate
4-benzyl-3-[1-(4-methylpyrimidine-5-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}piperidine-1-carboxylate
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methylpropyl)piperazine
N-[(4-methylphenyl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-[1-(4-methylpyrimidine-5-carbonyl)piperidine-4-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1-[(2S,4S)-1-(3-phenylpropyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carbonyl]azepane
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-5-methylpyrazine-2-carboxamide
1-(4-methoxyphenyl)-2,2-dimethyl-N-(thiophen-3-ylmethyl)cyclopropane-1-carboxamide
5-cyclopropanecarbonyl-1'-[(5-ethylpyridin-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
6-methyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
N-cyclopentyl-6-[3-(methoxymethyl)pyrrolidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(2R,6R)-4-(1-methyl-1H-pyrrole-2-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carbonyl]benzene-1,3-diol
3-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
5-cyclopropyl-1-{8-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
5-ethyl-2-(4-phenyl-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-imidazol-5-yl)pyridine
3-methyl-5-(3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}propyl)-4H-1,2,4-triazole
(1S,5R)-3-benzyl-6-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-phenyl-3-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepin-9-ylformamido}propanamide
1-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
3-(piperidin-3-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
1-[2-(methylsulfanyl)pyrimidin-4-yl]-N-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidin-4-amine
6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylpyrimidin-4-amine
N-(diphenylmethyl)-5-[(3-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
5-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}-2-methoxyphenol
N-[2-(4-phenylpiperidin-1-yl)ethyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(furan-2-ylmethyl)-N-methyl-1H-pyrazole-3-carboxamide
3-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
(4aS,7aR)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2-methoxyphenyl)-5-methyl-4-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]piperazin-2-one