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(3aS,6aS)-2-(cyclopropylmethyl)-5-[3-(1H-imidazol-1-yl)propanoyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-(2-hydroxyethyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-{2-[1-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
4-[2-(3-methoxyphenyl)piperidine-1-carbonyl]morpholine
4-[(2S)-3-hydroxy-2-methylpropyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-methyl-1-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}urea
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(1r,4r)-4-[5-(pentan-2-yl)-4-phenyl-1H-imidazol-1-yl]cyclohexan-1-ol
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
2-(cyclopropylmethyl)-9-{2-[4-(hydroxymethyl)phenyl]acetyl}-2,9-diazaspiro[5.5]undecan-3-one
4-[2-(5-acetylthiophen-3-yl)acetyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(5-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
2-butyl-8-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
(2S,4S)-N-ethyl-4-({[4-(methylsulfanyl)phenyl]methyl}amino)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1H-pyrazole-3-carboxamide
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-[(3-methylphenyl)methyl]-2-[4-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)morpholin-3-yl]acetamide
4-[3-(azepane-1-carbonyl)phenoxy]-N,N-dimethylpiperidine-1-sulfonamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1-(pyridin-2-yl)piperidine-3-carboxamide
2-[2-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-4-(pyrimidin-5-yl)phenoxy]acetic acid
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-(quinolin-4-ylmethyl)propanamide
1-{1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-4-yl}piperidin-4-ol
N-[2-(N-methylmethanesulfonamido)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methylacetamide
(1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-4-(2-phenoxyethyl)piperidin-4-yl)methanol
1-{[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-5-oxopyrrolidine-3-carboxylic acid
(1R,7S)-N-(1H-imidazol-2-ylmethyl)-3-(2-methoxyethyl)-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
8-(1,3-thiazol-2-ylmethyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
methyl 3-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}[3-(dimethylamino)propyl]carbamoyl)propanoate
2-(5-acetylthiophen-3-yl)-N-[(2,4,5-trifluorophenyl)methyl]acetamide
N-(1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-4-yl)methanesulfonamide
1-[2-(3-fluorophenyl)ethyl]-5-(morpholine-4-carbonyl)piperidin-2-one
N-{[4-(3-methoxyphenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]methyl}furan-2-carboxamide
1-methyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
[3-(1-methyl-1H-pyrazole-4-carbonyl)-9-(oxan-4-yl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
2-[4-(furan-3-carbonyl)morpholin-3-yl]-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]acetamide
N-(2-methylpropyl)-1-[1-(1H-pyrrol-2-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
N-(2-{1-[(4-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-3-methoxyphenyl)methyl]piperidin-4-yl}ethyl)acetamide
N-cyclobutyl-3-{[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]sulfamoyl}benzamide
1-[4-oxo-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(pyrrolidin-1-yl)ethane-1,2-dione
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
N-{[1-(2-acetylbenzoyl)piperidin-3-yl]methyl}-4-fluorobenzamide
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
5-[1-(3-methyl-2-oxopentanoyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-benzyl-1-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}piperidine-3-carboxamide
2-[4-({2-[2-(dimethylamino)ethyl]piperidin-1-yl}methyl)-3-methyl-1H-pyrazol-1-yl]ethan-1-ol
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)[(4-methyloxan-4-yl)methyl]amine
1-[1'-(1-ethylpyrrolidine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one