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N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
2-{3-[3-(4,6-dimethylpyrimidin-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-5-methylphenol
4-(1-butyl-1H-imidazol-2-yl)-1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidine
2-amino-6-(3-fluoro-4-methoxyphenyl)-4-(5-hydroxy-2-methoxyphenyl)pyridine-3-carbonitrile
8-[3-(2-methoxyphenyl)benzoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
(2S,4S)-4-amino-N,N-diethyl-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)pyrrolidine-2-carboxamide
2-(1H-1,3-benzodiazol-2-ylmethoxy)-1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
7-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]urea
5-methoxy-2-{[3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}phenol
8-{[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N3-cyclohexyl-1-cyclopentyl-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-{4-[3-(3-methylphenoxy)azetidin-1-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}pyridine
2-[4-(propan-2-yl)morpholin-2-yl]-N-(pyridin-2-ylmethyl)acetamide
(3aS,6aS)-2-ethyl-1-oxo-5-[3-(pyridin-2-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methyl]acetamide
2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
3-methyl-8-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
4-{4-[(6-chloropyridin-3-yl)methyl]piperazin-1-yl}-6-methoxypyrimidine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(2-fluorobenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-6-(morpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
5-(1H-indazol-1-yl)pyridine-3-carboxylic acid
6-[3-chloro-5-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
methyl 2-(4-{[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]amino}phenoxy)acetate
2-[5-(2-methylphenyl)-2H-1,2,3,4-tetrazol-2-yl]-N-(1-propyl-1H-indazol-3-yl)acetamide
ethyl 4-[(3-fluorophenyl)methyl]-1-(2-hydroxyethyl)piperidine-4-carboxylate
4-(hydroxymethyl)-1-[(7-methyl-2-phenyl-1H-indol-3-yl)methyl]piperidin-4-ol
3-cyano-5-fluoro-N-(oxan-3-ylmethyl)benzamide
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-3-[2-(morpholin-4-yl)propanoyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-{[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-4H-chromen-4-one
N-(4-{[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}phenyl)acetamide
5-chloro-2-[2-fluoro-6-(propan-2-yloxy)phenyl]pyrimidine
7-[(2,3-difluorophenyl)methyl]-2-(ethanesulfonyl)-2,7-diazaspiro[4.5]decane
4,5-dimethyl-3-({5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-2,3-dihydro-1,3-oxazol-2-one
2-[({2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
6-{3-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
2-(methylamino)-N-(3-methylphenyl)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidine-6-carboxamide
5-{2-[4-(3-chlorophenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-[2-(dimethylsulfamoyl)ethyl]-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
4-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-2,3,6-trimethylquinoline
3-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-4-phenyl-1H-pyrazol-5-amine
N,N-diethyl-4-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]benzamide
3-phenyl-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyrrolidin-3-ol
5-(4-methoxyphenyl)-3-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}-1,2,4-triazine
(3S,4S)-4-(4-fluorophenyl)-1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidin-3-ol
(2R,6S)-4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-2,6-dimethylmorpholine