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8-(5-chloro-3-fluoropyridin-2-yl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-(3-fluoro-4-methoxyphenyl)-3-[4-(pyridin-4-yl)piperidin-1-yl]-1,2,4-triazine
1-[2-(3-fluorophenyl)-1,3-benzoxazole-5-carbonyl]-4-phenylpiperidin-4-ol
2-(4-fluorophenyl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]morpholine
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-3-amine
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]propan-1-one
[5-({[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amino}methyl)furan-2-yl]methanol
N-[(3,4-difluorophenyl)methyl]-3-{1-[(2,3,6-trifluorophenyl)methyl]piperidin-3-yl}propanamide
4-(1-ethyl-1H-imidazol-2-yl)-1-(5-phenoxyfuran-2-carbonyl)piperidine
1-[1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]piperidin-3-ol
3-benzyl-4-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]piperazin-2-one
1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-2-methyl-1,4-diazepan-5-one
2-(3-methyl-1,2-oxazol-5-yl)-N-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]pyrrolidine-1-carboxamide
2-[({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)amino]pyridine-3-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-4-(1H-pyrazol-3-yl)benzamide
5-(5-chloro-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-2-(pyridin-3-yl)pyrimidin-4-ol
3-(1-benzyl-1H-imidazol-2-yl)-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-5-[(2-methylphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-{2-[(1,4-dioxan-2-ylmethyl)amino]pyrimidin-4-yl}-2-ethoxybenzoic acid
(4aR,8aR)-2-cyclopentanecarbonyl-7-[3-(pyridin-3-yl)propyl]-decahydro-2,7-naphthyridin-4a-ol
N-{[5-(methylcarbamoyl)furan-2-yl]methyl}-1-(oxan-4-yl)piperidine-3-carboxamide
1-ethyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-methanesulfonyl-1'-(5-methyl-1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-methyl-5-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1H-1,3-benzodiazole
3-(2-fluorophenyl)-N-[2-(morpholin-4-yl)ethyl]-3-phenylpropanamide
2-{2-methyl-7-oxo-6H,7H-pyrazolo[1,5-d][1,2,4]triazin-3-yl}-N,N-bis(propan-2-yl)benzamide
1-phenyl-N-{[4-({[3-(trifluoromethyl)phenyl]methyl}amino)quinazolin-2-yl]methyl}methanesulfonamide
4-methyl-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzamide
1-(diethylamino)-3-[4-({[(2,3-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
(2S)-1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
N-methyl-N-{[5-({6-oxo-2,7-diazaspiro[4.5]decan-2-yl}methyl)furan-2-yl]methyl}methanesulfonamide
1-[(1-ethylpyrrolidin-2-yl)methyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-{1'-[2-(3-fluorophenyl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
4-[3-(methoxymethyl)pyrrolidin-1-yl]-1-[3-(4-methylphenyl)phenyl]piperidine
5-chloro-2-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)phenol
2-[4-(8-methoxyquinolin-5-yl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
1-cyclopropyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-6-oxopiperidine-3-carboxamide
N-[(3S,7S,8aS)-3-[(4-chlorophenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,5-difluorobenzamide
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-methyl-2-(1-methyl-1H-indol-3-yl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
(3aS,6aS)-2-methanesulfonyl-5-[(3-methylpyridin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(azocan-1-yl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]acetamide
6-amino-1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]hexan-1-one
[(2S,6S)-4-[(2-butyl-1H-imidazol-4-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-3-(3-phenylpropyl)piperidin-3-yl)methanol
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-[1'-(3-chlorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-3-methylbut-2-en-1-one
5-cyclobutyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-1,3,4-oxadiazol-2-amine