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5-{2-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-2-methyl-3,4-dihydropyrimidin-4-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2,3-dihydro-1,4-benzodioxine-2-carboxamide
4-[(2-chloro-4-fluorophenyl)methyl]-3-[2-(4-cyclopentylpiperazin-1-yl)-2-oxoethyl]piperazin-2-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-3,3-diphenylpiperidine
4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]thiomorpholine
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
N,N-dimethyl-2-[(1S,5R)-3-(3-methylbenzenesulfonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
2-(azocan-1-yl)-1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
2-methoxy-1-{4-[5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-2-phenylethan-1-one
3-[5-(2,5-dimethylfuran-3-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
3-[(3-fluorophenyl)amino]-N-(2-phenylethyl)piperidine-1-carboxamide
(3R,4R)-1-(5-chloro-2-methylpyrimidine-4-carbonyl)-3-cyclopropyl-4-methylpyrrolidin-3-ol
1-[4-(4-methylphenoxy)piperidine-4-carbonyl]-4-(pyrrolidin-1-yl)piperidine
2-(5-fluoro-2-methylphenyl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carboxamide
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-amine
N-{1-[1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
4-(2,6-dimethylpyridin-3-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[2-(dimethylamino)ethyl]-N-methyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
N-(1-methyl-1H-indazol-3-yl)-2-{4-[6-methyl-2-(methylamino)pyrimidin-4-yl]-1H-pyrazol-1-yl}acetamide
3-[2-(methylsulfanyl)benzoyl]-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
N-{3-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-oxopropyl}acetamide
4-({1-[2-(morpholin-4-yl)acetyl]pyrrolidin-3-yl}methyl)benzoic acid
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-{3-[(4-fluorophenyl)methyl]piperidin-1-yl}ethan-1-one
8-(2-methoxybenzenesulfonyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-[2-({5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}amino)ethyl]-1,3,4-thiadiazol-2-amine
4-methyl-3-[({2-[(2R)-pyrrolidin-2-yl]ethyl}carbamoyl)amino]benzamide
2-methyl-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-1,8-naphthyridine-3-carboxamide
N-{[5-(cyclopentylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-methoxyacetamide
[2-(3,4-dimethoxyphenyl)ethyl](methyl)({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
2-(1-benzoylpiperidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 6-{3-tert-butyl-1-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}pyridine-2-carboxylate
7-(2,2-dimethylpropyl)-2-(6-methylpyridine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-4,6-dimethylpyrimidine
6-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carboxamide
6-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
4-[2-(3-hydroxyphenyl)-1H-imidazol-1-yl]-N-(2-methoxyethyl)-3-methylbenzamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
4-[3-(1H-pyrazol-3-yl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-2-amine
2-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-oxoethyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
1-[1-(3-phenylpropyl)piperidin-4-yl]-N-(prop-2-en-1-yl)piperidine-4-carboxamide
1-[2-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]-1,2-dihydropyridin-2-one
N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[1-(4-chlorophenyl)cyclobutyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
6-(4-acetylpiperazin-1-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
4-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-methoxy-6-({3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
4-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}-5-ethylfuran-2-carboxamide