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2-{[(4aS,7aR)-4-(2-carboxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-1,3-oxazole-4-carboxylic acid
4-(azocane-1-carbonyl)-2-(2-methylpyrimidin-5-yl)quinoline
N2,N2-diethyl-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidine-2,4-diamine
2-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidin-2-yl}pyridine
1-{2-[2-(3-fluorophenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(prop-2-en-1-yl)piperidine-3-carboxamide
4-[(5-acetylthiophen-3-yl)methyl]-1-(3-methoxyphenyl)-5-methylpiperazin-2-one
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-propanoylpiperidine-3-carboxamide
5-(oxane-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
(2-{[(5-ethylpyridin-2-yl)methyl][(5-methylthiophen-2-yl)methyl]amino}ethyl)dimethylamine
4-methyl-5-[1-(3-methylbutyl)-1H-pyrazol-4-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-ethyl-1-[4-(pyridin-3-yloxy)phenyl]urea
methyl 3-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidine-1-carbonyl]benzoate
N-[(4,6-dimethylpyridin-3-yl)methyl]-4-(piperidin-1-yl)butanamide
5-(6-chloro-2H-1,3-benzodioxol-5-yl)-1-cyclopentyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
9-(2-methoxypropanoyl)-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-ethoxy-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]benzamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-(oxolan-2-yl)thiophene-2-carboxamide
6-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-1,2-dihydropyridin-2-one
2-methyl-9-(2-methyl-2,3-dihydro-1-benzofuran-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(3-chlorophenyl)-3-oxo-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(5-methylthiophen-2-yl)methyl]pyrrolidin-3-yl]methanol
N2,6-dimethyl-N4-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)pyrimidine-2,4-diamine
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-ethyl-5-{[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyrimidin-2-amine
3-[3-(aminomethyl)pyrrolidine-1-carbonyl]-N-[(4-fluorophenyl)methyl]aniline
N-{1-[1-(2-cyclopentylacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
ethyl 1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(4-chlorophenyl)methyl]-4-(oxane-4-carbonyl)piperazine
4-[2-(2-fluorophenyl)ethyl]-3-(1-methyl-5-oxopyrrolidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)urea
4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-{[4-(methylsulfanyl)phenyl]methyl}piperidine
ethyl 3-{[(3S,4S)-3-(dimethylamino)-4-hydroxypyrrolidine-1-carbonyl]amino}-1-benzothiophene-2-carboxylate
4-(1-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)benzoic acid
5-cyclopropyl-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-oxazole-4-carboxamide
N-[3-(4-methyl-2-oxo-1,2-dihydroquinolin-3-yl)phenyl]acetamide
2-(4-methoxy-2-methylphenyl)-5-propylpyrimidine
1-amino-N-(2-{1-[(4-methylphenyl)methyl]piperidin-3-yl}ethyl)cyclobutane-1-carboxamide
(4aS,8aR)-6-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-({5-[(3-benzoylpiperidin-1-yl)methyl]furan-2-yl}methyl)-N-methylmethanesulfonamide
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine
ethyl 1-[(6-methylpyridin-2-yl)methyl]-3-(2-phenylethyl)piperidine-3-carboxylate
2-{6-[3-(morpholin-4-ylmethyl)phenyl]pyridin-3-yl}acetic acid
2-[5-(2,4-dimethoxyphenyl)-1,2,4-triazin-3-yl]-7-ethyl-2,7-diazaspiro[4.4]nonane
N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)oxolane-3-carboxamide
ethyl 2-{2-[(thian-4-yl)amino]ethyl}-1,3-thiazole-4-carboxylate
1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidine-3-carbonitrile
1-(cyclopropylmethyl)-N-ethyl-5-(1H-indol-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-ethyl-3-methyl-4-(4-oxo-4H-chromene-2-carbonyl)piperazin-2-one