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({5-[1-(1H-indole-2-carbonyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-[1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
3-(4-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)propanamide
4-[(4-methylphenyl)methyl]-3-[2-oxo-2-(4-phenylpiperidin-1-yl)ethyl]piperazin-2-one
1-[(3,5-dimethylphenyl)methyl]-4-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)piperazin-2-one
6-methyl-1-{3-oxo-3-[4-(pyridin-2-yl)piperazin-1-yl]propyl}-1,2-dihydropyridin-2-one
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-amine
(1S,5R)-6-propyl-3-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-3-(4-fluorophenoxymethyl)piperidine
N-ethyl-N-(2-hydroxyethyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(3,4-dichlorophenyl)-4-[(2-ethyl-1,3-thiazol-4-yl)methyl]morpholine
4-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-N,N-dimethylbenzamide
3-(4-chlorophenyl)-2-{[2-(hydroxymethyl)quinazolin-4-yl]amino}propan-1-ol
(3aR,6aS)-1-oxo-5-[(2-phenyl-1,3-oxazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazin-2-ol
1-[6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]azepane
[(2,2-dimethyloxan-4-yl)methyl](methyl)[(2-methylpyridin-4-yl)methyl]amine
[(6-methoxypyridin-3-yl)methyl](methyl)[1-(pyrimidin-4-yl)ethyl]amine
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-4,6-dimethylpyrimidin-2-amine
N-methyl-2-(morpholin-4-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
4-[3-(azepane-1-carbonyl)piperidin-1-yl]-2-[1-(thiophen-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-5-methoxy-1,4-dihydropyridin-4-one
1-(2,3-dihydro-1H-inden-2-yl)-4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
1-ethyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-{[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]amino}-N-(1,3-thiazol-2-yl)propanamide
5-[5-(methanesulfonylmethyl)pyridin-2-yl]-2-methylquinoline
3-methyl-8-(1-phenylcyclopentanecarbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3S)-3-(dimethylamino)azepan-1-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
1-(4-methoxyphenyl)-4-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidin-1-yl}butane-1,4-dione
8-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(4-{[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenoxy)ethan-1-ol
N-cyclopropyl-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2-(thiophen-3-yl)acetamide
N-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}oxan-4-amine
N-({1-[(3-fluoro-2,4-dimethylphenyl)methyl]piperidin-4-yl}methyl)-2-hydroxyacetamide
3-[1-(5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidin-4-yl]-1,3-oxazolidin-2-one
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
9-[(2,3-difluorophenyl)methyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
{1-[(4-methoxy-3-methylphenyl)methyl]-4-(2-phenoxyethyl)piperidin-4-yl}methanol
1-(cyclopropylmethyl)-3-[(2-methylphenyl)methyl]-6-(1H-pyrazol-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-2,3-dimethyl-N-(pyridin-2-ylmethyl)-1H-indole-5-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-(prop-2-ene-1-sulfonyl)piperidine-4-carboxylic acid
ethyl 4-{[6-(aminomethyl)-2-methylpyrimidin-4-yl]amino}piperidine-1-carboxylate
(2-{2-[1-(1,3-benzoxazol-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-[5-({[2-(1H-imidazol-4-yl)ethyl]carbamoyl}amino)-2-methylphenyl]-2-methylpropanamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
8-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(4aR,7aS)-1-cyclobutanecarbonyl-4-(1-methyl-1H-imidazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl){[5-(oxan-2-yl)furan-2-yl]methyl}amine
2-methyl-N-(pyridin-2-ylmethyl)-3-(1,2,3,6-tetrahydropyridine-1-carbonyl)aniline
ethyl 4-[9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidine-1-carboxylate