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3-(cyclopropylmethyl)-1-(2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carbonyl)piperidine-3-carboxylic acid
({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)({3-ethoxy-4-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-(pyridin-4-yl)propanamide
4-(5-methylpyridin-2-yl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidin-4-ol
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-methylpyrimidin-4-amine
N-(furan-2-ylmethyl)-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-amine
1-[(4-methanesulfonylphenyl)methyl]-3-(piperidin-1-ylmethyl)piperidine
3-hydroxy-1-[(3-methylphenyl)methyl]-3-{[(prop-2-en-1-yl)amino]methyl}piperidin-2-one
6-(6-methoxypyridin-3-yl)-2-(morpholin-4-yl)pyrimidin-4-amine
N-methyl-N-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(4H-1,2,4-triazol-4-yl)benzamide
N-[2-(furan-2-yl)ethyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
2-methoxy-4-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]quinoline
1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(pyridin-2-yl)piperazine
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
ethyl 2-[1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-2-yl]acetate
1-(pyridin-4-ylmethyl)-4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
5-{2-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(1,2-oxazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(5-cyano-1H-indol-1-yl)-N-(1-phenyl-1H-pyrazol-5-yl)acetamide
N-(propan-2-yl)-3-{5-[3-(pyridin-3-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
2-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-[3-(2-methoxyethoxy)phenyl]-3-[1-(pyridin-3-ylmethyl)piperidin-3-yl]urea
N-(2-methanesulfonamidoethyl)-5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl][(5-methylfuran-2-yl)methyl]amine
2-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-1-(pyridin-3-yl)ethan-1-ol
N-[(2,3-dimethoxyphenyl)methyl]-2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
(1R,2S,9R)-11-(3-phenyl-1,2,4-oxadiazol-5-yl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
2-(1-methylcyclopropanecarbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-{[(2-amino-5-ethyl-6-methylpyrimidin-4-yl)amino]methyl}-N,N-dimethylbenzamide
4-(1-hydroxy-2-phenylethyl)-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
2-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-7-propyl-2,7-diazaspiro[4.5]decan-6-one
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-methyl-N-(pyridin-4-ylmethyl)piperidin-4-amine
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-3-(pyridin-3-yl)propan-1-one
N-[(3-methoxyphenyl)methyl]-3-[1-(2-methylfuran-3-carbonyl)piperidin-3-yl]propanamide
4-[3-(benzyloxy)propyl]-6-methoxypyrimidine
(3S,4R)-4-(2-methoxyphenyl)-1-(4,4,4-trifluorobutanoyl)pyrrolidine-3-carboxylic acid
3-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-N-(thiophen-2-ylmethyl)propanamide
({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)(pyridin-2-ylmethyl)amine
4-(3,4-diethoxyphenyl)-2-propyl-1H-imidazole
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[(3,5-dichloropyridin-4-yl)methyl]-4-(pyridin-2-ylmethyl)piperazine
N-butyl-N-[(2E)-3-phenylprop-2-en-1-yl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
methyl 2-[(2,3-dihydro-1H-inden-5-yl)sulfamoyl]-6-(2,2-dimethylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[1-(hydroxymethyl)cyclopentyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-{[(butan-2-yl)(pyridin-4-ylmethyl)amino]methyl}benzonitrile
methyl 5-(5-ethyl-1,3-oxazole-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate