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1-{5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}piperidin-3-ol
(3S,4R)-1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
[(3R,4R)-1-(5-methyl-1,2-oxazole-4-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-4-(pyridin-2-ylmethyl)piperazine
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-5-fluoro-3,8-dimethylquinoline
4-cyclopentanecarbonyl-5-methyl-1-(4-methylphenyl)piperazin-2-one
(4aS,8aR)-1-[2-(5-methylfuran-2-yl)ethyl]-6-(1,2-oxazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-[2-(dimethylamino)-4-{[3-(pyridin-4-yl)propyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
4,6-dimethyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
(3R,4S)-4-{ethyl[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]amino}oxolan-3-ol
(3R,4R)-4-(azepan-1-yl)-1-[(8-chloroquinolin-2-yl)methyl]piperidin-3-ol
(2S,4R)-4-amino-N-ethyl-1-[2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetyl]pyrrolidine-2-carboxamide
(3R,4S)-1-(3-chloro-5-methoxybenzoyl)-4-cyclopropylpyrrolidin-3-amine
(3S,4R)-4-(2-methylphenyl)-1-(1,3-thiazol-2-ylmethyl)pyrrolidine-3-carboxylic acid
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-methylquinoline
1-ethyl-4-{[(1R,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-pyrrole-2-carbonitrile
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}benzamide
3-(3-chlorophenyl)-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-3-phenylpropanamide
3-(pyridin-3-yl)-4-(quinoxalin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-(2-{[3-(trimethyl-1H-pyrazol-1-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-2-(2-oxoimidazolidin-1-yl)acetamide
(3R,4R)-4-cyclobutyl-3-methyl-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-ol
1-(4-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}thiophen-2-yl)ethan-1-one
1-ethyl-8-[(1-methyl-1H-indol-3-yl)methyl]-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-fluoro-N-(3-{2-methoxy-4-[(3-methylpiperidin-1-yl)methyl]phenoxy}propyl)benzamide
dimethyl(2-{1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}ethyl)amine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3-(1-methyl-1H-imidazol-2-yl)piperidine
4-(1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-phenyl-1H-imidazol-5-yl)pyridine
5-(3-fluorophenoxymethyl)-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-pyrazole-3-carboxamide
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)quinoxalin-2-amine
4-[4-(1-ethoxyethyl)phenyl]-1-ethyl-1H-pyrazole
1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
(4aS,8aR)-6-[(2-methoxyphenyl)methyl]-1-methyl-decahydro-1,6-naphthyridine-4a-carboxylic acid
(3aR,5R,6S,7aS)-2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-octahydro-1H-isoindole-5,6-diol
2-(dimethyl-1,2-oxazol-4-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
N-tert-butyl-2-(1-methyl-1H-imidazol-2-yl)benzene-1-sulfonamide
1-cyclopropanecarbonyl-N-methyl-N-[1-(naphthalen-2-yl)ethyl]piperidin-4-amine
3-cyclobutyl-5-[(E)-2-[4-(trifluoromethyl)phenyl]ethenyl]-1H-1,2,4-triazole
N-cyclopropyl-2-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}acetamide
2-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-3-chloro-1H-indole
(1R,5R)-N,N-dimethyl-6-(1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-benzyl-8-(1,3-oxazole-4-carbonyl)-2,8-diazaspiro[5.5]undecane
2-[2-(1H-imidazol-1-ylmethyl)pyrrolidin-1-yl]-6-methylpyridine-3-carboxylic acid
N-(1-hydroxy-2-methylpropan-2-yl)-5-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(1,2-oxazole-3-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-(1-methyl-1H-pyrazol-4-yl)-4-(pyridin-4-yl)piperazine-1-carboxamide
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-2-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrimidine