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2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-(2-methoxyethyl)-N-[(3-methylthiophen-2-yl)methyl]acetamide
N-[3-(furan-2-yl)-3-phenylpropyl]piperidin-4-amine
2-[2-(dimethylamino)ethyl]-8-[4-(1H-pyrazol-4-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-2,7-dioxo-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-diazepane-4-carboxamide
4-(1,3-benzothiazol-6-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-acetyl-8-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[4-(3-fluorophenoxy)piperidin-1-yl]-3-(1H-imidazol-1-yl)butan-1-one
1-{4-[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-4-(4-fluorophenyl)butan-1-one
N-(2,4-dimethylphenyl)-3-{2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamido}propanamide
6-{methyl[(3-methylpyridin-2-yl)methyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
[(2,3-difluorophenyl)methyl]({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
(4aR,7aS)-1-cyclopropanecarbonyl-4-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(3-fluorophenyl)methyl]-4-{4-[2-(naphthalen-1-yl)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-2-(4-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
6-(diethylamino)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
4-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-1,4-diazepane-1-carbaldehyde
8-(2,6-dimethoxypyridine-3-carbonyl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
2-[3-benzyl-1-(3-methylphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methylacetamide
1-methyl-1-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-3-(prop-2-en-1-yl)urea
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}quinoline-2-carboxamide
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]benzamide
2-(2-methoxyphenoxy)-N-[(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]acetamide
3-methyl-1-(3-methylphenyl)-5-(2H-1,2,3-triazol-2-ylmethyl)-1H-1,2,4-triazole
3-[(3R,4S)-4-(dimethylamino)-1-[3-(pyridin-4-yl)propanoyl]piperidin-3-yl]propanoic acid
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-3-(1H-pyrazol-4-yl)propanamide
2,2,6,6-tetramethyl-4-(4H-1,2,4-triazol-4-yl)piperidine
N-(butan-2-yl)-1-ethyl-6-methyl-4-oxo-2-propyl-N-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
4-{2-[5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridine
4-[(2-methoxyphenyl)methyl]-3-{2-oxo-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethyl}piperazin-2-one
N-[(1S,2R)-2-(cyclooctylamino)cyclobutyl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-3,5,7-trimethyl-1H-indole
N-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-3-yl}-4-methyl-1,3-thiazol-2-amine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-3,4-dimethoxy-N-methylbenzamide
methyl 3-(furan-2-amido)-1-(3-methylbutyl)-5-[(oxan-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-(5,8-dimethoxy-4-methylquinolin-2-yl)-N-methylpyrrolidine-3-carboxamide
N-cyclopropyl-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine-2-carboxamide
5-[3-(aminomethyl)pyrrolidin-1-yl]-2-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-(3,4-dimethoxyphenyl)piperidin-3-amine
2-(2-methyl-1H-imidazol-1-yl)-1-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
2-[(2-carboxy-4,6-dimethoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
ethyl 1-{2-[4-(3-phenoxypropanamido)-1H-pyrazol-1-yl]acetyl}piperidine-2-carboxylate
3-(3-fluorophenyl)-N-[2-hydroxy-2-(pyridin-3-yl)ethyl]benzamide
1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-cyclopropyl-4-[(1,4-dioxan-2-ylmethyl)(methyl)sulfamoyl]benzamide
1-[3-(2-fluorophenoxy)azetidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1-(1H-imidazol-4-ylmethyl)-4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine
3-(1-methyl-1H-imidazol-2-yl)-6-[2-(piperidin-1-ylmethyl)phenoxy]pyridazine
1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
5-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidin-2-yl}-1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazole