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N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-2-fluoro-5-sulfamoylbenzamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
8-[(2S)-2-hydroxypropanoyl]-3-{3-[methyl(2-methylpropyl)amino]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]azocane
2-{[(3-methoxypropyl)(1-methylpiperidin-4-yl)amino]methyl}benzonitrile
4-(2H-1,3-benzodioxol-4-ylmethyl)-2-[(4-fluorophenyl)methyl]morpholine
8-(3-hydroxy-4-methylbenzoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N2,N2,5,6-tetramethyl-N4-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)pyrimidine-2,4-diamine
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-7-fluoro-2-oxo-1,2-dihydroquinoline-4-carboxamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-5-cyclopropyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1-methyl-1H-indole-3-carboxamide
1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-[(3-methoxyphenyl)methyl]-N-(pyridin-4-ylmethyl)piperidin-3-amine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-1,3-oxazole-4-carboxamide
1,2-dimethyl-4-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazine
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]{[4-(trifluoromethoxy)phenyl]methyl}amine
1-[2-(3-chlorophenyl)ethyl]-4-[(1H-imidazol-2-ylmethyl)amino]pyrrolidin-2-one
N-methyl-3-propyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
N-cyclopropyl-1-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
4-[5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
2-phenoxy-N-{2-[7-(quinolin-4-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}acetamide
(2R,4S)-4-hydroxy-1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperidine-2-carboxylic acid
8-chloro-2-({[2-(pyrrolidine-1-sulfonyl)ethyl]amino}methyl)quinolin-4-ol
2-({4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}methyl)benzoic acid
1-(3-carbamoylpyridin-2-yl)-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylic acid
3-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea
2-[4-(4-methylquinolin-2-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
5-methyl-N-[1-(oxan-4-yl)piperidin-4-yl]-1-propyl-1H-pyrazole-4-carboxamide
N-({1-[(3-ethyl-1,2-oxazol-5-yl)methyl]pyrrolidin-3-yl}methyl)-3-hydroxy-2-methylbenzamide
4-{2-[(5-methyl-4-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}pyrimidin-2-yl)sulfanyl]ethyl}morpholine
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-methoxy-4-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]pyridine-3-carbonitrile
2-[1-(3-methylbut-2-en-1-yl)-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl]ethan-1-ol
N-cyclohexyl-N-methyl-1-{2-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carboxamide
2-[cyclopentyl(methyl)amino]-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
(2S,4R)-4-(2-ethoxyacetamido)-N,N-diethyl-1-(furan-3-carbonyl)pyrrolidine-2-carboxamide
5-ethyl-1'-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(5-propyl-1,3,4-oxadiazol-2-yl)-4-[2-(pyrrolidin-1-yl)ethyl]piperidine
3-(furan-2-yl)-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3-phenylpropanamide
N-[(2S,4R,6S)-2-benzyl-6-(1,3-thiazol-2-yl)oxan-4-yl]acetamide
3-methyl-7-[2-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-oxoethyl]-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
(3S,4R)-4-(2-methoxyphenyl)-1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]pyrrolidine-3-carboxylic acid
1-(3-{3-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]phenyl}-1H-pyrazol-1-yl)propan-2-ol
[4-({3-[(2-chloro-6-fluorophenyl)methoxy]phenyl}methyl)morpholin-3-yl]methanol
3-(1H-1,2,3-benzotriazol-1-yl)-1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}propan-1-one
1-[2-(dimethylamino)-6-(trifluoromethyl)pyrimidin-4-yl]-4-(hydroxymethyl)azepan-4-ol
3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N-(pyrimidin-4-ylmethyl)benzamide
3-[1-(3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoyl)piperidin-4-yl]-1,3-oxazolidin-2-one
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-(4-chloro-1H-pyrazol-1-yl)propan-1-one
2-(2-methoxyethyl)-8-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one