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N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}furan-3-carboxamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(propan-2-yl)piperidin-4-yl]methyl}acetamide
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2,3-dihydro-1,4-benzodioxine-6-sulfonamide
[(3R,4S)-1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
2-ethyl-8-(6-fluoro-4-hydroxyquinoline-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-methyl-N-{[2-(3-methylphenyl)-6-oxo-1,6-dihydropyrimidin-4-yl]methyl}piperazine-1-sulfonamide
N-({1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)-3-methylbenzamide
(1R,3s,6r,8S)-4-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)-4-azatricyclo[4.3.1.13,8]undecane
4-(hydroxymethyl)-1-[(4-methanesulfonylphenyl)methyl]piperidin-4-ol
5-[5-(3,5-dimethylbenzenesulfonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]-1,2-oxazole
N-[(4-fluorophenyl)methyl]-2-(2H-indazol-2-yl)acetamide
(3aS,6aS)-5-(6-methyl-2-phenylpyrimidin-4-yl)-1-oxo-2-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S)-2-{[3-(3-hydroxy-3-methylbutyl)phenyl]formamido}-3-methylbutanamide
3-methanesulfonamido-N-phenyl-5-[({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}amino)methyl]benzamide
[(2S,6S)-4-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
(1R,5R)-3-(2-chloro-3-methylbenzoyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-6-(cyclobutylmethyl)-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(furan-2-ylmethyl)-2-methanesulfonyl-N-(3-methylbutan-2-yl)acetamide
N,7,8-trimethyl-2-(1H-pyrazol-4-yl)-N-[2-(pyrrolidin-1-yl)ethyl]quinoline-4-carboxamide
N-[3-(4-methoxyphenyl)propyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
ethyl 1-(5-acetylthiophene-2-carbonyl)-3-[(3-chlorophenyl)methyl]piperidine-3-carboxylate
1-cyclopentyl-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-N-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[1-(furan-2-yl)ethyl]-6-(4-methoxyphenyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-[(4-hydroxyphenyl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3S,5S)-5-[(4-fluorophenyl)carbamoyl]-1-(1H-imidazol-2-ylmethyl)piperidine-3-carboxylic acid
2-methyl-N-{[5-(methylsulfanyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,3-thiazole-4-carboxamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-4-(1H-1,2,4-triazol-1-yl)butanamide
(1R,3S)-3-(2-hydroxyethoxy)-7-[(2E)-3-phenylprop-2-en-1-yl]-7-azaspiro[3.5]nonan-1-ol
3-(2,5-dimethoxyphenyl)-1-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1-methylurea
1-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-4-(hydroxymethyl)piperidin-4-ol
2-(2-methyl-1H-indol-3-yl)-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}ethan-1-one
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4-sulfamoylbenzamide
1-(2,6-difluorobenzoyl)-3-[2-(4-fluorophenyl)ethyl]piperidine
(3S,4R)-1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
4-(3,3-dimethylpyrrolidine-1-carbonyl)-2-(2-ethylpyrimidin-5-yl)-7-fluoroquinoline
2-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1,2,3,4-tetrahydroisoquinoline
N3-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-N5-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
5-methyl-3-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-indazole
2-(4-fluorophenyl)-N-(2-{7-[3-(5-methylfuran-2-yl)butyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-7-(2-methoxyacetamido)-N-methyl-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
5-ethyl-2-[3-(2-methoxyphenoxy)azetidin-1-yl]pyrimidine
3-{1-[3-(dimethylamino)pyrazin-2-yl]piperidin-4-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-ethyl-9-[(3-fluoro-4-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
5-[3-hydroxy-3-(2-methylphenyl)pyrrolidine-1-carbonyl]-2-(thiophen-2-yl)pyrimidin-4-ol
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-3-(naphthalene-1-carbonyl)piperidine
4-[4-(2,5-dihydro-1H-pyrrol-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-yl]pyridine
N,N-dimethyl-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carboxamide
1-[6-(furan-3-yl)pyridazin-3-yl]azepane