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[4-benzyl-1-(9-methyl-9H-carbazole-3-carbonyl)piperidin-4-yl]methanol
1-(2-methyl-1-benzofuran-7-carbonyl)-3-[(methylsulfanyl)methyl]piperidine
(4aS,8aR)-6-(1,3-thiazol-4-ylmethyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[(3-chloro-4-methoxyphenyl)methyl]-N-methylpiperidine-2-carboxamide
2-ethoxy-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
6-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{[2-(1H-1,3-benzodiazol-2-yl)ethyl](methyl)amino}pyrazine-2-carbonitrile
2-amino-6-cyclopentyl-4-[2-(2-hydroxyethoxy)phenyl]pyridine-3-carbonitrile
(3S,5R,9R)-5-hydroxy-11-[(4-methylphenyl)methyl]-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
N-methyl-N-(propan-2-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,3,5-trimethyl-1H-indole-2-carboxamide
7-fluoro-2-methyl-N-{1-oxaspiro[4.4]nonan-3-yl}quinoline-4-carboxamide
1-[(3-fluorophenyl)methyl]-4-(5-methoxypyrimidin-2-yl)piperazin-2-one
1-[(2-fluorophenyl)methyl]-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1H-imidazol-5-yl)methyl]amine
7-(2-methoxyethyl)-2-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
11-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]-7-thia-2,5-diazatricyclo[6.4.0.02,6]dodeca-1(12),5,8,10-tetraene
8-methoxy-2-[4-phenyl-1-(piperidin-4-yl)-1H-imidazol-5-yl]quinoline
2-[4-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)phenyl]-6-(methoxymethyl)-3,4-dihydropyrimidin-4-one
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)morpholine-2-carboxamide
1-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]hex-5-yn-1-one
1-(2-methanesulfonylethyl)-2-[4-(trifluoromethyl)phenyl]-1H-imidazole
8-(5-methyl-1,2-oxazole-3-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
{4-[({[5-(2-chlorophenyl)furan-2-yl]methyl}(methyl)amino)methyl]oxan-4-yl}methanol
{1-[(4-chloro-2-fluorophenyl)methyl]-3-(cyclopropylmethyl)piperidin-3-yl}methanol
N-methyl-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]-N-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
2-amino-4-(4-methyl-1H-imidazol-5-yl)-6-[4-(morpholin-4-ylmethyl)thiophen-2-yl]pyridine-3-carbonitrile
4-methoxy-3-{[3-(3-methoxyphenoxymethyl)piperidin-1-yl]methyl}phenol
4-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-1-phenyl-1H-1,2,3-triazole
2-({1-[1-(pyridin-2-yl)piperidine-3-carbonyl]piperidin-4-yl}oxy)pyrimidine
N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-4-methoxybenzamide
6-methyl-N4-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}pyrimidine-2,4-diamine
1-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-oxoethyl}-2-methyl-1,4-dihydroquinolin-4-one
8-(pent-4-enoyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
ethyl 1-(4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzoyl)piperidine-4-carboxylate
5-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)-6-methyl-2-(1H-pyrazole-4-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
2-[(6-amino-2-methylpyrimidin-4-yl)amino]-N,N-dimethylethane-1-sulfonamide
N-methyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]acetamide
N-(diphenylmethyl)-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
N-[2-(1H-indol-3-yl)ethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[7-methyl-2-(morpholin-4-yl)quinolin-3-yl]methyl}amine
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
4-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-6-ethyl-N,N-dimethylpyrimidin-2-amine
N,5-dimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyrazine-2-carboxamide
4-(dimethylamino)-N-(3-methoxy-4-methylphenyl)azepane-1-carboxamide
3-(4-{4-[(dimethylamino)methyl]thiophen-2-yl}-1H-1,2,3-triazol-1-yl)propane-1,2-diol
1-cyano-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)cyclopropane-1-carboxamide
1-[2-(2-chloro-6-methoxyphenyl)pyridine-4-carbonyl]-4-methylpiperazine
6-(4-ethylphenyl)-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide