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N-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
5-[(2-ethyl-4-methyl-1H-imidazol-1-yl)methyl]-3-(phenoxymethyl)-1,2,4-oxadiazole
2-[4-(4-fluorophenyl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-1-[2-(pyridin-3-yl)piperidin-1-yl]ethan-1-one
(4S)-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-4-phenyl-1,3-oxazolidin-2-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}propanamide
6-(3-chlorophenyl)-7-(cyclopropylmethyl)-2-(3-hydroxyazetidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
5-methyl-3-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-2-(4H-1,2,4-triazol-4-yl)pyridine
N-(adamantan-2-ylmethyl)-6-({4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
8-(2-methyl-2,3-dihydro-1-benzofuran-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
[1-(1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}piperidin-4-yl)ethyl]dimethylamine
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N,2-dimethyl-4-phenyl-1,3-thiazole-5-carboxamide
2-(cyclopent-1-en-1-yl)-1-[7-(hydroxymethyl)-9-methyl-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-one
2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)acetamide
4-({[(2-amino-1,3-thiazol-4-yl)methyl]amino}methyl)-2-chloro-6-ethoxyphenyl acetate
2-(3-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
3-[(4-cyclobutyl-6-methylpyrimidin-2-yl)amino]-2,2-dimethylpropan-1-ol
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(pyrrolidin-1-yl)piperidine
6-[(3-methoxyphenyl)methoxy]-4-(2-methylpropanoyl)-1-(2-phenylethyl)-1,4-diazepan-2-one
(2R,3R,6R)-3-phenyl-5-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(2-hydroxyethyl)-2-(pyridin-4-yl)-N-(1,3-thiazol-2-ylmethyl)pyrimidine-5-carboxamide
6-chloro-2-{[1-(2-methylpyridin-4-yl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
2-cyclopropyl-8-[(2-fluoro-4-methoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(oxolane-2-carbonyl)-4-[4-(pyridin-3-yl)pyrimidin-2-yl]-1,4-diazepane
(2S)-2-amino-1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-5-hydroxypyridine-2-carboxamide
2-(1-benzofuran-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
methyl (2S,4R)-1-[(6,7-dimethyl-2-oxo-2H-chromen-4-yl)methyl]-4-hydroxypyrrolidine-2-carboxylate
3-phenyl-7-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N'1-[(2-methoxyphenyl)methyl]-N'1-[(3-methylphenyl)methyl]cyclopropane-1,1-dicarboxamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3-phenoxypropanamide
4-(2-fluorophenoxy)-1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
6-ethyl-4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-methylquinoline
N-[2-(diethylamino)ethyl]-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-N,5-dimethyl-1H-pyrazole-4-carboxamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-(oxan-4-yl)piperidin-4-amine
N-[(3S,4R)-1-(2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
2-(propan-2-yloxy)-1-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-1-one
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}pyridine-4-carboxamide
2-(3-hydroxypropyl)-9-[2-(methylamino)-2-phenylacetyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}pyridine
N-[(1-ethylcyclopropyl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
{9-cyclopropanecarbonyl-3-[(2-methyl-1H-imidazol-4-yl)methyl]-3,9-diazaspiro[5.5]undecan-1-yl}methanol
(3S,4S)-4-({[(2-chloro-6-fluorophenyl)methyl]amino}methyl)piperidin-3-ol
2-[(2-chlorophenyl)methyl]-4-(1,5-dimethyl-1H-pyrazole-3-carbonyl)morpholine
1-(3-methanesulfonamido-4-methoxyphenyl)-3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}urea
(2S)-N2-[2-(cyclohex-1-en-1-yl)ethyl]-N2-[(4-fluorophenyl)methyl]pyrrolidine-1,2-dicarboxamide
1-{2-[4-(4,6-dimethoxypyrimidin-2-yl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
N-[(3R,4R)-4-hydroxypyrrolidin-3-yl]-3,5,7-trimethyl-1H-indole-2-carboxamide
N-[(3R,4R)-1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
1-[(2-fluorophenyl)methyl]-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide