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1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-(4-fluorophenyl)piperidine
2-({5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propan-1-ol
2-(1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-imidazol-2-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole
1-(3-methoxyphenyl)-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-one
3-hydroxy-3-{[(1-phenylcyclopropyl)amino]methyl}-1-(2-phenylethyl)piperidin-2-one
3-{2-[(2,1,3-benzothiadiazol-5-ylmethyl)amino]propyl}-3,4-dihydroquinazolin-4-one
1-(adamantan-2-ylmethyl)-5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)pyrrolidin-2-one
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(2-methyl-1,3-benzoxazole-6-carbonyl)pyrrolidin-3-yl]methanol
4-ethyl-6-[4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazin-1-yl]pyrimidine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-ethyl-1H-pyrazole-4-carboxamide
N-{2-[ethyl(3-methylphenyl)amino]ethyl}-2-(trifluoromethyl)pyrimidin-4-amine
N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[4-(3-methoxyphenyl)benzoyl]pyrrolidin-3-yl]methanol
ethyl 1-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxylate
3-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1,2-dihydroquinolin-2-one
{3-[(4-fluorophenyl)methyl]-1-[(4-methylphenyl)methyl]piperidin-3-yl}methanol
5-(4-methyl-1,4-diazepan-1-yl)-2-(1,3-thiazol-2-ylmethyl)-2,3-dihydropyridazin-3-one
2-(diethylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-2-(oxan-4-yl)ethan-1-one
9-(2-methoxyethyl)-1-methyl-4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
5-chloro-3-methyl-2-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}-1H-indole
2-chloro-4-(1-{3-[(1-methylpiperidin-4-yl)oxy]propyl}-1H-imidazol-2-yl)phenol
1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
7-[(2,3-dimethoxyphenyl)methyl]-2-(pyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4,5-dimethyl-6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-(3-hydroxypropyl)-N-(pyridin-4-ylmethyl)quinoxaline-6-carboxamide
4-phenyl-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidine-4-carbonitrile
6-(2,5-dimethylfuran-3-yl)-2-(3-{[4-(methylamino)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N,N-diethyl-2-{[2-oxo-1-(2-phenylethyl)-4-(pyridin-3-ylmethyl)-1,4-diazepan-6-yl]oxy}acetamide
[(3R,4S)-4-(morpholin-4-ylmethyl)-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]methanol
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
4-methyl-2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}pyrimidine
2-[(2-{4-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}ethyl)sulfanyl]pyridine
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2,5-dimethoxybenzamide
2-(4-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-[4-({[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenyl]-2-methylbut-3-yn-2-ol
1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-(1,4-dioxan-2-ylmethyl)-3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)sulfonyl]benzamide
(4aR,8aS)-1-[(4-methoxyphenyl)methyl]-6-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-(2-chlorophenyl)-3-[1-(1,3-oxazole-5-carbonyl)piperidin-4-yl]propanamide
1-[1-(cyclopropanesulfonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)morpholine-4-carboxamide
4-{4-[1-(1-benzothiophen-5-ylmethyl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}piperidine
2-amino-6-cyclopropanecarbonyl-4-[4-(2-hydroxyethoxy)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(4-methylphenyl)-4-[(1-oxo-1λ4-thian-4-yl)amino]pyrrolidin-2-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-ethyl-1,2-oxazole-5-carboxamide
(2S,4R)-4-amino-1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
2,3-dimethyl-6-[1-(propan-2-yl)piperidine-3-carbonyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
2-(2,5-dimethylphenoxy)-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-{1-oxaspiro[4.4]nonan-3-yl}urea