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2-{[4-(4-methylphenyl)-5-(1H-pyrazol-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-methylpyridazin-3-amine
N2,N4-dimethyl-N2-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidine-2,4-diamine
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(propan-2-ylsulfanyl)ethan-1-one
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]thian-4-amine
2-(4-{1-[2-(benzenesulfonyl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)pyridine
(1S,6R)-9-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
N-[(2-methoxynaphthalen-1-yl)methyl]-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
N-[(3-chlorophenyl)methyl]-5-cyclopropyl-N-methyl-1,3,4-oxadiazol-2-amine
N,N-diethyl-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
7-(3-phenyl-1,2,4-oxadiazol-5-yl)-2,7-diazaspiro[4.4]nonane-1,3-dione
3-{[(3S,4R)-3-acetamido-4-propylpyrrolidin-1-yl]sulfonyl}-4-fluorobenzoic acid
6-(azepan-1-ylmethyl)-N-(9H-fluoren-9-yl)-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
2-{1-[1-(1H-imidazole-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-N-[1-(thiophen-2-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
4-(2-methoxypyridin-3-yl)-5,6-dimethyl-2-(trifluoromethyl)pyrimidine
dimethyl({[6-(6-methylquinolin-3-yl)pyridin-3-yl]methyl})amine
(4aS,7aR)-1-(6-methoxy-1-methyl-1H-indole-2-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(1-benzylpiperidin-4-yl)-N-(cyclopropylmethyl)-N-propylpiperidine-3-carboxamide
2-(2-methylphenyl)-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]acetamide
1-[2-(dimethylamino)-4-({[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}amino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-[2-(1H-imidazol-1-yl)ethyl]-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine
3-[(4-fluorophenyl)formamido]-N-[(3S)-2-oxoazepan-3-yl]propanamide
(2S,4S)-4-[4-(4-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}phenyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
N-(carbamoylmethyl)-2-[1-(4-chlorophenyl)-3-(furan-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
N-(cyclohexylmethyl)-3-[(oxan-4-yl)sulfamoyl]benzamide
1-[(2,5-dimethoxyphenyl)methyl]-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
1-(4-methylphenyl)-4-[2-(pyrazin-2-yl)acetyl]piperazin-2-one
2-cyclohexyl-N-(2-oxooxolan-3-yl)-1,3-benzoxazole-6-carboxamide
(1S,5R)-6-(2-methoxypyridine-4-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-[(3R,4S)-1-(2-hydroxyethyl)-4-propylpyrrolidin-3-yl]-5-(hydroxymethyl)furan-2-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-(5-chlorothiophene-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-[(2-chlorophenyl)methyl]-3-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-3-yl}propanamide
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-5-(morpholin-4-ylmethyl)furan-3-carboxamide
3-{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-4-yl}phenol
1-methanesulfonyl-4-[3-(5-methylfuran-2-yl)benzoyl]-1,4-diazepane
2-[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-decahydro-2,7-naphthyridine-2-sulfonamide
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidine-1-carboxamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(quinoline-2-carbonyl)pyrrolidin-3-yl]methanol
(4aR,7aS)-1-(pyridin-4-ylmethyl)-4-(1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}benzonitrile
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(2-oxopiperidin-1-yl)butanamide
4-[(dimethylamino)methyl]-1-[(5-propylfuran-2-yl)methyl]azepan-4-ol
N-[2-(dimethylamino)ethyl]-N,1-dimethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-ethyl-N-[2-(2-fluorophenoxy)ethyl]-2-(propan-2-yloxy)acetamide