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N-{imidazo[1,2-a]pyrazin-3-ylmethyl}-2H-1,3-benzodioxole-5-carboxamide
(2S,4R)-N,N-diethyl-4-(2-hydroxyacetamido)-1-[(5-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(quinoxalin-2-yl)pyrrolidin-3-yl]methanol
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
3-[(1-{5-[(dimethylamino)methyl]furan-2-carbonyl}piperidin-4-yl)methyl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
6-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]pyridin-3-ol
(1R,7S)-3-[4-(2-hydroxyethyl)phenyl]-N-methyl-4-oxo-N-(pyridin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-[2-(4-fluorophenyl)-2-hydroxyacetyl]-1-(4-methoxyphenyl)piperazin-2-one
7-chloro-N-[5-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
5-amino-N-benzyl-N-(prop-2-en-1-yl)-1H-pyrazole-3-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-methyl-N-(thian-4-yl)acetamide
4-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-1-(pyridin-4-yl)ethyl]morpholine
3-[(1-acetylpiperidin-4-yl)oxy]-N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-methoxybenzamide
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,6-dichlorophenyl)urea
N-{3,4-dihydrospiro[1-benzopyran-2,1'-cyclohexane]-4-yl}-6-oxo-1,6-dihydropyridine-2-carboxamide
6-[3-chloro-5-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
4-(5-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
7-(cyclopropylmethyl)-2-(2-ethylpyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[3-(trifluoromethyl)pyridin-2-yl]-decahydro-1,6-naphthyridin-2-one
5-({4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-2-(methylsulfanyl)pyrimidine
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(diethylamino)ethan-1-one
3-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]-N-[(3,4-difluorophenyl)methyl]propanamide
1-(2-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-3-methoxy-1,2-dihydropyridin-2-one
methyl 4-[5-methyl-4-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)-1,3-oxazol-2-yl]benzoate
N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-4-(1H-1,2,4-triazol-1-yl)butanamide
N2,N2-dimethyl-6-({[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)-1,3,5-triazine-2,4-diamine
2-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-1,3-thiazole-4-carboxamide
3-(1-methyl-1H-pyrazol-5-yl)-N-(piperidin-3-ylmethyl)propanamide
1-[1-(1,2,3,4-tetrahydroisoquinoline-6-carbonyl)piperidin-4-yl]piperidin-4-ol
N-(cyclohex-1-en-1-ylmethyl)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
4-(2,6-dimethylpyridin-3-yl)-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]pyrimidin-2-amine
3-[(7-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine
(1S,5R)-3-[(2,4-difluorophenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{4-[(hexan-3-yl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
(3S,4S)-4-cyclopropyl-1-(1-methyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxylic acid
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-4-oxo-N-[(3S)-2-oxoazepan-3-yl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1'-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-oxo-3-(pentan-3-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
3-(3-fluoro-4-methoxyphenyl)-4-(1H-imidazol-2-yl)-1-(2-methylphenyl)-1H-pyrazole
2-(5-{[cyclopentyl(methyl)amino]methyl}-1-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl)acetamide
1-(4-chloro-3-fluorobenzoyl)-N-(3,4-dimethoxyphenyl)piperidin-3-amine
1-(4-{methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}piperidin-1-yl)ethan-1-one
3-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1-{4-[(trifluoromethyl)sulfanyl]phenyl}urea
N-(2,3-dihydro-1H-inden-4-yl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carboxamide
1-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidin-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
(4aR,7aS)-1-(furan-2-carbonyl)-4-[(2E)-3-phenylprop-2-en-1-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(1R,2S)-2-phenylcyclopropyl]-1H-pyrazole-3-carboxamide
N-(3,4-difluorophenyl)-1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-amine