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3-(2-fluorophenyl)-N-[2-(2-methylpropanesulfonyl)ethyl]-1H-pyrazole-4-carboxamide
4-(piperidin-1-yl)-1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]piperazine
2-benzyl-9-(pent-2-yn-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
1-[(4-fluorophenyl)methyl]-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]ethan-1-one
4-methyl-N-(2-{4-[(4-phenylpiperazin-1-yl)methyl]phenoxy}propyl)benzamide
1-{4-[3-(1H-pyrazol-3-yl)phenyl]benzoyl}piperidine
ethyl 4-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylate
ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)(isoquinolin-5-ylmethyl)amine
2-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)-N-[2-(N-methylmethanesulfonamido)ethyl]acetamide
1-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
2,7,8-trimethyl-4-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]quinoline
N-cyclopentyl-3-(3-methyl-1H-pyrazol-1-yl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)propanamide
(4aS,8aS)-2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)-decahydro-2,7-naphthyridin-4a-ol
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidine-4-carboxylic acid
4-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-1,3-thiazole
(4S)-4-hydroxy-N-(4-methoxy-2-methylphenyl)-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carboxamide
1'-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N4-[(3-chlorophenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
1-[(3-fluorophenyl)methyl]-4-[(3R,4R)-1-methyl-4-(2-methyl-1H-imidazol-5-yl)pyrrolidine-3-carbonyl]piperazine
1-(2,4-dichloro-3-methylphenyl)-3-[2-(N-methylmethanesulfonamido)ethyl]urea
6-(2-fluoro-4-methoxyphenyl)-2-(3-hydroxyazetidine-1-carbonyl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
4-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidine
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1H-1,3-benzodiazole-5-carboxamide
2-[1-(1-methylpiperidin-4-yl)-4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
5-chloro-4,6-dimethyl-3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-(cyclopropylmethyl)-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[3-(2-ethoxyethoxy)benzoyl]-4-(pyrrolidine-1-carbonyl)piperidine
{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
3-(pyridin-3-yl)-1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)propan-1-one
4-(oxane-4-carbonyl)-2-(2-phenylethyl)morpholine
2-{1-[(5-methylfuran-2-yl)methyl]-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-yl}ethan-1-ol
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-methylphenyl)methyl]piperidine
(2S,4R)-4-(2,5-dimethylfuran-3-amido)-N-ethyl-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
(2S)-1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidine-2-carboxamide
8-(3-chloro-5-methoxybenzoyl)-2,8-diazaspiro[4.5]decan-3-one
(1S,5R)-3,6-bis(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(1-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
4-ethoxy-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]pyrimidin-2-amine
6-[1-(2,3-dihydro-1H-inden-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
1-ethyl-6-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}-1H-indole
3-[(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)methyl]piperidine
N-[(4-ethylphenyl)methyl]-N,2-dimethyl-4-phenylpyridine-3-carboxamide
(2S,4S)-N-ethyl-4-(2-hydroxyacetamido)-1-{[(thiophen-2-ylmethyl)carbamoyl]methyl}pyrrolidine-2-carboxamide
(2S,4S)-4-amino-N-ethyl-1-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxamide
[3-(2-phenylethyl)piperidin-3-yl]methanol
5-[(4-benzylpiperidin-1-yl)methyl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
5-(1,2,3,4-tetrahydronaphthalen-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine