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1-[2-chloro-5-(morpholine-4-carbonyl)phenyl]-3-[2-(pyrrolidin-1-yl)ethyl]urea
2-acetyl-8-(1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N,1,3-trimethyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-(2-oxo-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)-1,2-dihydropyridin-2-one
2-amino-6-(4-methoxyphenyl)-4-{2-[(propan-2-yl)amino]pyrimidin-5-yl}pyridine-3-carbonitrile
N-(3-hydroxypropyl)-N-methyl-3-(piperidin-4-ylmethyl)benzamide
7-fluoro-2-(1-methyl-1H-pyrazol-4-yl)-4-(morpholine-4-carbonyl)quinoline
3-[2-(phenylamino)pyrimidine-5-carbonyl]-3,9-diazaspiro[5.6]dodecan-10-one
N-[2-(dimethylamino)ethyl]-N,1-dimethyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N'1-[2-(pyridin-3-yloxy)propyl]cyclopropane-1,1-dicarboxamide
3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-8-(1-methoxypropan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(1-methyl-1H-pyrazole-5-carbonyl)-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
3-[(3R,4S)-4-(morpholin-4-yl)-1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperidin-3-yl]propan-1-ol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,2-dimethyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-[2-(1H-imidazol-1-yl)propyl]-2,6,8-trimethylquinoline-4-carboxamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-4-(1H-1,2,4-triazol-1-yl)butanamide
5-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-2-methyl-3,4-dihydropyrimidin-4-one
4-(benzyloxy)-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine
3-[4-(2-methoxyacetamido)-1H-pyrazol-1-yl]-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]benzamide
N-[(1-hydroxycyclohexyl)methyl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
3-(2H-1,3-benzodioxol-5-yl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
4-[5-(5-phenyl-1,2-oxazol-3-yl)-1,2,4-oxadiazol-3-yl]pyridine
[(4-fluorophenyl)methyl](pyridin-4-ylmethyl){[6-(trifluoromethyl)pyridin-3-yl]methyl}amine
5-({[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]amino}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-[2-({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]benzene-1-sulfonamide
4-(1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)pyridine
3-cyclopropyl-1-(4-methanesulfonylphenyl)-3-[(5-methylthiophen-2-yl)methyl]urea
5-{[2-(1H-indol-3-yl)ethyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
ethyl 2-[benzyl({2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl})amino]acetate
13-(4-hydroxy-3,5-dimethoxyphenyl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
2-ethyl-5-{2-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-6-methyl-3,4-dihydropyrimidin-4-one
2-ethoxy-1-(7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
9-[(3-methoxyphenyl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(dimethylamino)methyl]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1,3-thiazole-4-carboxamide
1,3,6-trimethyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
5-{2-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-methyl-2-(morpholin-4-yl)propyl]-4-(1H-pyrazol-4-yl)butanamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-1-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
1'-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
4-(1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carbonyl)morpholine
(2R,3R,6R)-5-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-hydroxy-2-methyl-N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)pyrimidine-5-carboxamide
4-[(2-methylpyrimidin-5-yl)methyl]-2-(3-phenylpropyl)morpholine
2-benzyl-9-[2-(oxolan-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(4-fluorophenyl)methyl]-N-[3-(1H-imidazol-1-yl)propyl]-5-(2-methoxyacetamido)-1H-1,3-benzodiazole-7-carboxamide
3-{[3-(methoxymethyl)piperidin-1-yl]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)propan-1-one
N-(4-{1-[(1-methylpiperidin-2-yl)methyl]-1H-imidazol-2-yl}phenyl)acetamide
(2S,4S)-4-amino-1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-N-ethylpyrrolidine-2-carboxamide