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(3S,4R)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
3-[4-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)-1H-pyrazol-1-yl]propanoic acid
(4aR,8aR)-7-(2,1,3-benzoxadiazol-4-ylmethyl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
5-(2,4-difluoro-3-methoxybenzoyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-{4-chloro-2-[1-(oxolan-3-yl)-4-phenyl-1H-imidazol-5-yl]phenoxy}acetamide
4-{1-[1-(4-methyl-1H-imidazole-2-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
5,6-dimethyl-2-(4-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
ethyl 1-[2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]piperidine-3-carboxylate
5-{[3-(methoxymethyl)piperidin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
3-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-1-[4-(furan-2-yl)phenyl]-3-methylurea
3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-N,N-dimethylpiperidine-1-sulfonamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(piperidin-4-yl)acetamide
N-[(2-chlorophenyl)methyl]-2-(ethylamino)-N-(prop-2-en-1-yl)pyrimidine-5-carboxamide
5-(2-chlorobenzoyl)-1-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{6-[(1S,3R)-1-[2-(dimethylamino)ethoxy]-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]pyridin-3-yl}ethan-1-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-3-phenylprop-2-ynamide
N-[2-(1H-indol-3-yl)ethyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
(2S,4S)-1-(2,5-dimethylfuran-3-carbonyl)-N,N-diethyl-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(1R,2R)-2-hydroxycyclohexyl]-N-propylbenzamide
2-methyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3,6-dimethyl-N-(propan-2-yl)-2-(1-propyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
4-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-1,3,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidine
2-[4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
4-(4-fluorophenyl)-1-(2-methyl-1-benzofuran-5-carbonyl)-1,2,3,6-tetrahydropyridine
6-oxo-1-[2-(pyridin-2-yl)ethyl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidine-3-carboxamide
3-[1-(2-hydroxypyridine-3-carbonyl)piperidin-3-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(4-ethylpiperazin-1-yl)-1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]ethan-1-one
1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-4-(pyridin-4-yl)piperazine
3-{4-[(dimethylamino)methyl]-4-hydroxyazepane-1-carbonyl}-1,6-dimethyl-1,4-dihydroquinolin-4-one
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amine
3-(naphthalene-1-carbonyl)-9-(oxan-4-yl)-3,9-diazaspiro[5.5]undecane
4-{1-[1,3-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}morpholine
3-[(2-chlorophenyl)methyl]-5-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(2-hydroxyphenyl)acetamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylcyclopentanecarboxamide
ethyl 1-[(3-hydroxyphenyl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
4-({2-[2-(dimethylamino)pyrimidin-5-yl]-1H-imidazol-1-yl}methyl)benzene-1-sulfonamide
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(furan-2-ylmethyl)amine
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
2-(3-hydroxypiperidin-1-yl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
1-cyclopentyl-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(3S,4R)-1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
N-(2-{4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}-2-oxoethyl)-2-methylpropanamide
(2R,3R)-3-[3,5-bis(propan-2-yl)-1H-pyrazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1,3-dimethyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-[(dimethylamino)methyl]-2-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}pyrimidin-4-amine
2-(4-methyl-6-{4-[(oxan-2-ylmethyl)amino]piperidin-1-yl}pyrimidin-2-yl)phenol
2-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
4-(1H-1,3-benzodiazol-1-yl)-1-[(5-methylthiophen-2-yl)methyl]piperidine-4-carboxylic acid