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N-(2-methoxyethyl)-3,5-dimethyl-N-[(5-methylthiophen-2-yl)methyl]-1H-indole-2-carboxamide
3-{4-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1,3-thiazol-2-yl}pyridine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
5-{[(8-methoxy-4-methylquinolin-2-yl)amino]methyl}pyrrolidin-2-one
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,2,5-thiadiazole-3-carboxamide
N-[(2-fluorophenyl)methyl]-4-(4-{[1-(trimethyl-1H-pyrazol-4-yl)ethyl]amino}piperidin-1-yl)benzamide
2-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-6-(4H-1,2,4-triazol-4-yl)pyridine
1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
(4aR,8aS)-1-{[4-(trifluoromethyl)phenyl]methyl}-6-(3,4,5-trimethoxybenzoyl)-decahydro-1,6-naphthyridin-2-one
7-fluoro-2-methyl-4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}quinoline
2-(dimethylamino)-4-methyl-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]pyrimidine-5-carboxamide
2-ethyl-6-methyl-1-[(5-methylfuran-2-yl)methyl]-3-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}-1,4-dihydropyridin-4-one
6-[2-(pyrrolidine-1-sulfonyl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-[3-(dimethylamino)propyl]-5-[(4-fluorophenyl)methyl]-5-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-2-(2-methyl-1H-imidazol-1-yl)acetamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-2-(pyrrolidin-3-yl)benzamide
4-({1-[(1s,4s)-4-hydroxycyclohexanecarbonyl]pyrrolidin-3-yl}methyl)benzoic acid
2-(4-methoxyphenyl)-N-(4-{4-[(pyridin-4-ylmethyl)amino]piperidin-1-yl}phenyl)acetamide
3-[(dimethylamino)methyl]-1-[3-(hydroxymethyl)-8-methylquinolin-2-yl]pyrrolidin-3-ol
1-[2-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)-2-oxoethyl]imidazolidine-2,4-dione
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
1-(cyclohexylmethyl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-(4-methoxyphenoxy)-1-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperidine
(3R,5S)-N-[3-(1H-imidazol-2-yl)propyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
4-[2-(4-acetylphenoxy)acetyl]-1-(2-methylphenyl)piperazin-2-one
1-[2-(dimethylamino)ethyl]-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
1-(4-methoxyphenyl)-4-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}butane-1,4-dione
2-{1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(5-hydroxypyrazine-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
(4aS,7aR)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(2S,6S)-4-[(2-aminopyridin-3-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
(1R,5R)-6-[(2-fluoro-4-methoxyphenyl)methyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(4aS,8aR)-6-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
4-methyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]benzene-1-sulfonamide
N'-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N'-methyl-N-(2-methylphenyl)propanediamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-3-ol
N-[(2-ethoxypyridin-3-yl)methyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
3-(1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-N-(oxolan-2-ylmethyl)propanamide
2-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-oxo-N-phenylacetamide
(3R,4S)-4-cyclopropyl-1-[2-(2-phenylethoxy)benzoyl]pyrrolidin-3-amine
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N,N-dimethyl-5-{[2-(2-phenylethyl)morpholin-4-yl]methyl}-1,3-thiazol-2-amine
4-[2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-1-hydroxyethyl]phenol
7-(1H-indole-7-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{4-[2-(morpholin-4-yl)ethyl]piperazin-1-yl}propan-1-one
1-[(3-methoxyphenyl)methyl]-4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
ethyl 2-(N-methyl-1-{2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-4-yl}formamido)acetate
N-[(4-acetamidophenyl)methyl]-2-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]acetamide