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(1-methyl-1H-imidazol-2-yl)(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-4-yl)methanol
N6-benzyl-N5-(1,4-dioxan-2-ylmethyl)-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-amine
6-cyclopentyl-1-methyl-4-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-1H-pyrazolo[3,4-d]pyrimidine
2-methyl-N-[2-(pyridin-3-yloxy)propyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl){[4-(pyrimidin-2-yloxy)phenyl]methyl}amine
6,7-dimethoxy-2-[1-(1-methyl-1H-indole-2-carbonyl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
3-{2-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}azepan-2-one
(3R,5S)-N-[(3,4-dimethoxyphenyl)methyl]-5-(morpholin-4-ylmethyl)-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
2-(2-{9-oxa-2-azaspiro[5.5]undecan-2-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
1'-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-[1-(3,5-dimethyl-1H-indole-2-carbonyl)piperidin-3-yl]-1,3-benzoxazole
4-{4-[(3,4-dihydro-2H-1-benzopyran-3-yl)amino]piperidin-1-yl}-6-methylpyrimidin-2-amine
N-(adamantan-2-yl)-6-{[benzyl(ethyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(2-fluorophenyl)propan-1-one
2-[5-(1-cyclopentyl-5-oxopyrrolidin-3-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(3,4-dimethylphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(2-{[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-yl]formamido}ethyl)-1,3-thiazole-4-carboxylic acid
N-methyl-2-(methylsulfanyl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]benzamide
5-(methoxymethyl)-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl][(4-methoxyphenyl)methyl](pyridin-2-ylmethyl)amine
7-hydroxy-4-{2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}-1,2,3,4-tetrahydroquinolin-2-one
5-(2-fluorophenoxymethyl)-N-methyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-3-carboxamide
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}oxan-4-amine
N-(2-fluorophenyl)-3-{1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl}propanamide
3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]-1-[4-(pyridin-4-yl)piperazin-1-yl]propan-1-one
2-(1H-1,3-benzodiazol-2-ylmethoxy)-N-methyl-N-(pyrazin-2-ylmethyl)acetamide
5-methoxy-9-[4-(1H-pyrazol-3-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecane
3-(2,5-dihydro-1H-pyrrole-1-carbonyl)-5-(3-fluorophenoxymethyl)-1H-pyrazole
1-benzyl-3-(2-methoxyethyl)-8-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(3-chlorophenyl)-1-[4-(2-hydroxyethyl)piperazin-1-yl]-3-phenylpropan-1-one
5-ethyl-2-methyl-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]pyrimidin-4-amine
N-cyclopropyl-2-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-4-carboxamide
2-(3-chlorophenyl)-N-[4-(4-{[3-(1H-pyrazol-1-yl)propyl]amino}piperidin-1-yl)phenyl]acetamide
N-[(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-N-methylmethanesulfonamide
4-(3-ethyl-1,2-oxazole-5-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
3-cyclohexyl-N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
[(3R,4R)-1-[(6-chloroquinolin-2-yl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-methyl-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]pyrazine-2-carboxamide
1-(2-fluorophenyl)-3-(oxan-4-yl)-5-[2-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole
5-{[(2,3-difluorophenyl)methyl]amino}-1-methyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(4aR,8aS)-1-(5-fluoro-1H-indole-2-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
({5-[1-(1H-1,2,3-benzotriazole-5-carbonyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-methyl-6-oxo-N-(pyridin-3-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
4-(1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)-1λ6-thiomorpholine-1,1-dione
methyl 3-(oxolane-2-amido)-1-(2-phenylethyl)-5-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{octahydropyrrolo[1,2-a]piperazin-2-yl}-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridine
N-phenyl-4-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}piperidine-1-carboxamide
N-(3-cyclopentylpropyl)-N-methyl-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
(1R,2R,4R)-N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)bicyclo[2.2.1]hept-5-ene-2-carboxamide