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[(3R,4R)-1-[2-(dimethylamino)benzoyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
5-chloro-3-methyl-N-{[4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-1H-indole-2-carboxamide
ethyl 4-(8-methyl-3-{[N-(oxolan-2-ylmethyl)-1-1,3-thiazol-5-ylformamido]methyl}quinolin-2-yl)piperazine-1-carboxylate
2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-1,3-thiazole-4-carboxamide
5-[2-(piperidin-1-yl)ethyl]-7-{[(pyridin-3-ylmethyl)amino]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-butyl-N-(furan-2-ylmethyl)-2-methyl-5-sulfamoylbenzamide
N-cyclopropyl-N-(1H-indol-5-ylmethyl)-2-(1H-pyrazol-1-yl)butanamide
[2-(1H-1,3-benzodiazol-2-yl)ethyl][1-(3-methoxyphenyl)propan-2-yl]amine
1-methyl-3-(1-methylpiperidin-3-yl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(2E)-3-(pyridin-3-yl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}prop-2-en-1-one
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-3-(2-methoxyphenyl)propanamide
1-[2-({[4-methoxy-3-(methoxymethyl)phenyl]methyl}(methyl)amino)ethyl]piperidin-2-one
N-[(3-fluorophenyl)methyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
2-amino-6-tert-butyl-4-(3-hydroxyphenyl)pyridine-3-carbonitrile
4-(2-methyl-1H-imidazol-1-yl)-1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}butan-1-one
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]acetamide
1-{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}azetidin-3-ol
methyl 4-(5-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
2-amino-3-ethyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-cyclopentyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
4-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-3-ethyl-1-methylpiperazin-2-one
4-(ethylamino)-N,5-dimethyl-N-(thiophen-3-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
1-(3-chlorophenyl)-4-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl}piperazine
(4aR,7aS)-1-(cyclopropylmethyl)-4-(3,4-dimethoxybenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methyl-3-oxo-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
N'-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-methyl-N'-(oxolan-2-ylmethyl)ethanediamide
1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-(2-phenylethyl)piperidine-3-carboxamide
4-(2H-1,3-benzodioxol-5-ylmethyl)-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[3-(pyridin-4-yl)propanoyl]-1λ6-thiomorpholine-1,1-dione
1-(carbamoylmethyl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidine-3-carboxamide
3-[4-(2-methoxyethoxy)phenyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
2-(4-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperazin-1-yl)pyrimidine
2-benzyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1,3-thiazole-4-carboxamide
(4aS,8aR)-1-(2-methylpropyl)-6-[3-(pyrazin-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
5-cyclohexaneamido-N-[1-(4-fluorophenyl)ethyl]-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-3-propylpiperidine-3-carboxylic acid
1-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-3-[1-(propan-2-yl)-1H-pyrazol-4-yl]urea
2-(2-methoxyethyl)-9-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
4-methoxy-1-(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzoyl)piperidine
1-({4-methyl-5-[1-(6-methylpyridazin-3-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
2-[4-({methyl[(3-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-1-(4-methylpiperidin-1-yl)ethan-1-one
3-{[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]amino}-1λ6-thiolane-1,1-dione
6-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}quinoline
2-{4-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}-4-(2-methoxyphenyl)pyrimidine
1-(2-cyclohexylethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-(5,6,7,8-tetrahydronaphthalen-1-yl)urea
1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-3-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}urea
{[2-(furan-2-yl)pyrimidin-5-yl]methyl}(methyl){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-(4-methylphenyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole