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2-[4-(4-aminopyrimidin-2-yl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl]acetic acid
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-(1H-imidazol-4-yl)-1-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1H-imidazole
[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
5-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-5-oxopentanamide
2,2-dimethyl-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
3-{imidazo[1,2-a]pyridin-2-yl}-1-{1-oxa-8-azaspiro[4.6]undecan-8-yl}propan-1-one
N-(adamantan-2-ylmethyl)-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N,N-dimethylpiperidine-3-carboxamide
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-[(propylamino)methyl]piperidin-2-one
2-(5-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
2-{[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}-3-methoxyphenol
4-ethyl-3-{1-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(1H-1,3-benzodiazol-1-yl)-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidine-4-carboxylic acid
methyl (2S)-1-[4-(1H-1,2,4-triazol-5-yl)benzoyl]pyrrolidine-2-carboxylate
N,N,5-trimethyl-2-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrimidin-4-amine
3-cyclobutyl-4-[2-(4-methoxyphenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(2-chlorophenoxy)ethyl]pyridine-4-carboxamide
3-phenyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-3-(pyridin-2-yl)propanamide
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-(propan-2-yl)pyrimidin-4-amine
(3R,5S)-5-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrrolidin-3-ol
6-{4-[2-(dimethylamino)-2-(3-methylphenyl)acetyl]piperazin-1-yl}pyridine-3-carbonitrile
N-[(3S,4R)-1-(3-chlorothiophene-2-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
N-(1-methylcyclohexyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-{4-[4-(cyclopentylamino)-5-methylthieno[2,3-d]pyrimidine-6-carbonyl]piperazin-1-yl}-1λ6-thiolane-1,1-dione
4-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-1,4-oxazepan-6-ol
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(2-methylprop-2-en-1-yl)acetamide
methyl N-{2-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-2-oxoethyl}carbamate
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-2-(methylsulfanyl)pyridine-3-carboxamide
(4aS,8aR)-6-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-1,9-dioxaspiro[5.5]undecan-4-amine
(3S,4S)-4-cyclopropyl-1-[2-(2-methoxyphenoxy)-2-methylpropanoyl]pyrrolidine-3-carboxylic acid
N-methyl-5-(oxolan-2-yl)-N-[2-(phenylsulfanyl)ethyl]thiophene-2-carboxamide
1-[1-(1-benzothiophene-2-carbonyl)piperidin-3-yl]-4-(2-methoxyphenyl)piperazine
4-[5-(2-methylpropyl)thiophen-2-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-methyl-4-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-2-hydroxy-N-(oxolan-2-ylmethyl)acetamide
1-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-1-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]butan-1-one
N-[2-(1H-indol-3-yl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
dimethyl({4-methyl-5-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(1-methyl-1H-pyrazol-3-yl)acetamide
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(2-methoxyethyl)(propan-2-yl)amine
methyl 2-(diethylsulfamoyl)-6-(2-fluorobenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(1-benzyl-1H-pyrazol-5-yl)-1-[1-(furan-2-ylmethyl)piperidin-4-yl]urea
(3R,4S)-4-propyl-1-[4-(trifluoromethyl)benzenesulfonyl]pyrrolidin-3-amine
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
4-{2-[2-(thiomorpholin-4-ylmethyl)phenoxy]ethyl}morpholine
2-{2-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one
5-[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]piperidin-2-one