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N-(3-hydroxypropyl)-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
2-(cyclohex-1-ene-1-carbonyl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
1-(3-{5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)-2-(thiophen-3-yl)ethan-1-one
ethyl 4-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazine-1-carboxylate
1-[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]-4-(4-chlorophenyl)piperidin-4-ol
1-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3-(2-methoxyphenyl)propan-1-one
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(4-methoxyphenyl)ethyl]acetamide
1-{3-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
2-amino-4-(6-ethoxypyridin-3-yl)-6-(trimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-benzyl-N-cyclopropyl-4-oxo-5-(4-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-[1-(1-cyclopentanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-3-phenylpropanamide
N-ethyl-3,5,7-trimethyl-N-(propan-2-yl)-1H-indole-2-carboxamide
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(6-methoxynaphthalen-2-yl)-4-[2-(pyridin-2-yl)ethyl]morpholine
2-methyl-3-[4-(2-methylphenoxy)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indol-4-one
1-(1-ethylpiperidin-4-yl)-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
6-{pyrazolo[1,5-a]pyridin-7-yl}pyridine-2-carbonitrile
3,5-dimethyl-2-({[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}methyl)pyridin-4-ol
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide
3-(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
2-(4-chloro-2-methylphenoxy)-1-{4-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidin-1-yl}propan-1-one
2-methyl-3-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-6H,7H-pyrazolo[1,5-d][1,2,4]triazin-7-one
2-[2-(dimethylamino)ethyl]-8-[2-(methylamino)pyrimidine-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[(2-chlorophenyl)methyl]-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
6-chloro-2-(1-ethyl-1H-pyrazol-4-yl)-N-methyl-N-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]quinoline-4-carboxamide
N-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}-2-(4-phenylphenyl)acetamide
(4aS,8aR)-6-[2-(2-methoxyphenoxy)ethyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-({1-[3-(methylsulfanyl)propyl]piperidin-3-yl}methyl)naphthalene-1-carboxamide
1-(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
1-{2-[({5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}amino)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}ethan-1-one
1-(4-chlorobenzoyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N-ethyl-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-N-(pyridin-4-ylmethyl)piperidin-3-amine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}furan-3-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-{3-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-oxopropyl}pyrrolidin-2-one
1-[5-(4-methoxyphenyl)furan-2-carbonyl]-4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
N-{[7-(1H-indole-5-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-sulfonamide
2-(2H-1,3-benzodioxol-5-yl)-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}acetamide
3-butanamido-N-{2-[(pyridin-3-yl)amino]ethyl}benzamide
[(3R,4R)-1-(2,3-dichlorobenzoyl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
1-methyl-N-[1-(methylcarbamoyl)cyclohexyl]-2-oxo-1,2-dihydroquinoline-3-carboxamide
1-{1-[(2-cyanophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
N'-{2-[4-(1-benzofuran-5-ylmethyl)morpholin-2-yl]ethyl}ethanediamide
(3S,5S)-1-(2-cyclopentylacetyl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
3-(furan-2-yl)-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
N-[(2,3-dimethoxyphenyl)methyl]-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1S,2S)-2-{5-[4-(2-hydroxyethoxy)phenyl]-4-phenyl-1H-imidazol-1-yl}cyclohexan-1-ol
2-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]benzonitrile
N-cyclohexyl-N-methyl-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
2-(2-hydroxyethyl)-9-(2-phenylpropyl)-2,9-diazaspiro[5.5]undecan-3-one