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N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(2-methylpropyl)piperidin-4-amine
2-(1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}pyrrolidin-2-yl)-1,3-thiazole
2-(4-{1,9-dioxaspiro[5.5]undecan-4-yl}piperazin-1-yl)pyrimidine
4-(2-chlorobenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
(2S)-2-amino-1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-6-hydroxyhexan-1-one
1-[2-(oxolan-3-yl)ethyl]-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
4-(4-chlorophenyl)-1-[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]butan-1-one
1-(4-methyl-3-phenylpiperazin-1-yl)-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
1-(1-cycloheptylpiperidin-3-yl)-3-[2-(trifluoromethyl)phenyl]urea
methyl({[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
2-{2-methyl-2,7-diazaspiro[4.5]decan-7-yl}propane-1,3-diol
1-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
N-ethyl-2-(2-oxo-1,2-dihydroquinoxalin-1-yl)-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][(1-methylpiperidin-3-yl)methyl](2-phenylethyl)amine
3-(4H-1,2,4-triazol-4-yl)naphthalen-2-ol
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
3-(1-methyl-1H-imidazole-2-carbonyl)-1-[2-(methylsulfanyl)benzoyl]piperidine
2-ethyl-8-[(4-fluorophenyl)methanesulfonyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[2-methyl-2-(morpholin-4-yl)propyl]-2,7-diazaspiro[4.5]decane
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
2-{4-[3-methoxy-5-(trifluoromethyl)phenyl]-3,5-dimethyl-1H-pyrazol-1-yl}acetamide
1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
3-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)-N-(6-methylpyridazin-3-yl)benzamide
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]furan-3-carboxamide
6-{4-[4-(cyclohexylmethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-9H-purine
7-[(2,6-dimethoxyphenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-(4-fluorophenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
1-(3-chlorophenyl)-4-[1-(1-ethylpiperidin-4-yl)piperidin-3-yl]piperazine
(1,3-benzothiazol-2-ylmethyl)({[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
3-(2-fluorophenyl)-5-(5-methoxyfuran-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-(2-methyl-1H-indol-3-yl)ethan-1-one
2-(dimethyl-1,3-thiazol-5-yl)-1-[4-(3-methylphenoxy)piperidin-1-yl]ethan-1-one
(1R,2s,3S,6R,7r,8S)-N-(2H-1,3-benzodioxol-5-ylmethyl)-11,12-dioxatetracyclo[6.2.1.13,6.02,7]dodecane-2-carboxamide
N-[1-(1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-4-yl)-1H-pyrazol-5-yl]pyridine-3-carboxamide
3-[(4aR,7aS)-4-[(5-cyano-1H-pyrrol-3-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
2-(1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)ethan-1-amine
[4-(2-phenylethyl)-1-(thian-4-yl)piperidin-4-yl]methanol
5-ethyl-4-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyrimidine
3-{5-[(2R)-2-amino-2-cyclohexylacetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-(propan-2-yl)propanamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-5-methoxy-1,2-dimethyl-1H-indole-3-carboxamide
1-{4-[5-phenyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}-2-(1,3-thiazol-4-yl)ethan-1-one
N-(1H-imidazol-2-ylmethyl)-5-(methoxymethyl)-N-methyl-1,3,4-oxadiazole-2-carboxamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-(3,3,5,5-tetramethylcyclohexyl)propanamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-[3-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
3-(2-{3-[3-(4-benzylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
3-(furan-2-yl)-3-{[3-(2-hydroxyphenyl)-1H-pyrazol-5-yl]formamido}propanoic acid
methyl[(1-methyl-1H-pyrazol-4-yl)methyl]({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
N-(2,2-dimethylpropyl)-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine