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methyl (2S)-2-{[2-(dimethylamino)-2,3-dihydro-1H-inden-2-yl]formamido}-3-phenylpropanoate
4-(5-ethyl-1,3,4-oxadiazol-2-yl)-N,N-dimethylpiperazine-1-carboxamide
2-[(3-{ethyl[(1-methyl-1H-imidazol-2-yl)methyl]carbamoyl}phenyl)amino]acetic acid
3-(5-chloro-2-methoxybenzoyl)-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidine
(1R,2S,9R)-11-{[2-(propylamino)pyrimidin-5-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
2-(6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
6-[3-(hydroxymethyl)pyrrolidin-1-yl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
N-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
3-[1-(3-methylpyridin-2-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydroquinoxalin-2-one
2-(methylamino)-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]pyrimidine-5-carboxamide
2-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyrimidin-4-amine
2-{4-[2,5-dioxo-4-(2-phenylethyl)imidazolidin-4-yl]piperidin-1-yl}pyridine-3-carboxamide
1-(3-chloro-2-ethoxyphenyl)-3-[3-(1H-imidazol-2-yl)propyl]urea
N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-amino-N-[2-(benzyloxy)ethyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-{4-phenyl-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}propan-1-ol
2-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,3-dihydro-1,2-benzothiazol-3-one
1-(2,6-dimethylpyridin-4-yl)-4-[4-(pyrrolidin-1-yl)benzoyl]piperazine
4-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-(2-methyl-1-benzofuran-5-yl)benzamide
3-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)methyl]pyridin-2-amine
4-({4-[(3,3-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}methyl)-1-(1H-pyrazole-4-carbonyl)piperidine
N-[2-(4-ethoxyphenyl)ethyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
(2S,4R)-4-amino-N-ethyl-1-(1H-indol-4-ylmethyl)pyrrolidine-2-carboxamide
2-{5-[1-(cyclohexylmethyl)-1H-1,2,4-triazol-5-yl]-1H-pyrazol-3-yl}phenol
N-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]-2-(dimethyl-1,2-oxazol-4-yl)acetamide
1-ethyl-5-[3-(3-ethylphenoxy)azetidine-1-carbonyl]piperidin-2-one
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
N-[(1-methylpiperidin-2-yl)methyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-(oxan-4-yl)-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-{[2-(2-fluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}-2-methoxyphenol
methyl 6-(cyclopent-1-ene-1-carbonyl)-2-{[(4-fluorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-ethyl-3,5-difluoro-N-[2-(4-methoxyphenoxy)ethyl]pyridine-2-carboxamide
5-(4-hydroxypiperidine-1-carbonyl)-1-(3-phenylpropyl)piperidin-2-one
(3R,4R)-1-{5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3-methyl-4-(oxan-4-yl)piperidin-4-ol
(1S,5R)-3-(2,5-dimethylfuran-3-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-(1,2,3,4-tetrahydronaphthalen-1-yl)benzamide
N-cyclopropyl-3-fluoro-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)benzamide
6-chloro-2-methyl-N-[2-(N-methylmethanesulfonamido)ethyl]imidazo[1,2-a]pyridine-3-carboxamide
2-methyl-N-(oxolan-2-ylmethyl)-N-propyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
4-{4-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]piperazin-1-yl}butan-1-ol
5-chloro-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[(2R,3R)-2-methoxy-1'-(pyridin-2-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-[1-cyclopentyl-7-(4-formyl-1,4-diazepane-1-carbonyl)-1H-1,3-benzodiazol-5-yl]benzamide
5-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-3-[(4-fluorophenyl)methyl]-5-methylimidazolidine-2,4-dione
5-ethyl-N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-1,3-oxazole-4-carboxamide
ethyl 4-(6-{[3-(2-methylphenyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carbonyl)piperazine-1-carboxylate
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-3-methoxybenzamide
2-(4-{[2-(morpholin-4-yl)ethyl]amino}piperidin-1-yl)pyridine-4-carbonitrile
methyl 3-[(3S,4R)-1-[(2,5-dimethylphenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoate