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1-[4-(pyridin-2-yl)piperazin-1-yl]-3-{1-[(2,3,6-trifluorophenyl)methyl]piperidin-3-yl}propan-1-one
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-(1-methylpiperidin-3-yl)urea
(2R,3R)-3-{[2-(2-chlorophenoxy)ethyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[4-(1H-indol-2-yl)phenyl]-1-(oxane-2-carbonyl)piperidine-4-carboxamide
(4R)-3-methyl-N-[(2-propyl-1,3-thiazol-4-yl)methyl]-1,3-thiazolidine-4-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-methyl-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
methyl 2-[({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)carbamoyl]benzoate
3-(2,5-dioxoimidazolidin-4-yl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}propanamide
2-fluoro-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-5-sulfamoylbenzamide
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-2,4-difluoro-3-methoxy-N-methylbenzamide
2-{4-[2-(methylsulfanyl)benzoyl]-2-oxopiperazin-1-yl}benzonitrile
3-{[1-(4-fluorophenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
ethyl 4-{1-[1-(ethoxycarbonyl)piperidin-4-yl]piperidin-3-yl}piperazine-1-carboxylate
ethyl 4-[(4-{[1-(2-chlorobenzenesulfonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
4,5-dimethyl 1-[(3S,5S)-1-(cyclohexylmethyl)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-3-(morpholin-4-yl)propanamide
4-[2-(dimethylamino)phenyl]-6-methylpyrimidin-2-amine
1-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-cyclopentyl-N-[2-(1H-indol-1-yl)ethyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
N-[4-(5-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)phenyl]acetamide
5-(4-hydroxypiperidin-1-yl)-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-N-cyclohexyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
7-(2,2-dimethylpropyl)-2-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
1-{2-[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]propyl}-3,5-dimethyl-1H-pyrazole
(3aS,6aR)-5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-3-methyl-2-phenylbutanamide
(2S,4S)-4-{4-[(adamantan-1-ylformamido)methyl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxylic acid
N-[(4-hydroxyazepan-4-yl)methyl]-1-methyl-3-phenyl-1H-thieno[2,3-c]pyrazole-5-carboxamide
(1-{[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)methanol
N-(1-cyclopropylethyl)-2-(methylsulfanyl)pyridine-3-carboxamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2,4-dimethylpyrimidine-5-carboxamide
N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-[1-(furan-2-yl)ethyl]-5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
4-(4-chlorophenyl)-N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}butanamide
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-4-(1H-pyrazol-4-yl)butanamide
2-[1-cyclohexyl-5-(5-methyl-1,2-oxazol-3-yl)-1H-1,2,4-triazol-3-yl]pyridine
1-[2-(3-fluorophenyl)ethyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
N-(adamantan-2-ylmethyl)-1-ethyl-3-(4-methylpiperazine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[4-({[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amino}methyl)phenyl]but-3-yn-1-ol
methyl 4-[2-(piperazin-1-ylmethyl)phenyl]benzoate
N-(butan-2-yl)-2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-(3-phenylprop-2-yn-1-yl)acetamide
4-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyrrolidin-2-one
N-methyl-5-(1-{[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
4-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
5-[(dimethylsulfamoyl)amino]-N,1-dimethyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-(2-methylpropyl)-1H-1,3-benzodiazole-7-carboxamide
3-[2-(2-fluorophenyl)ethyl]-1-[5-(methoxymethyl)furan-2-carbonyl]piperidine
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-[(4-fluorophenyl)methyl]-5-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazole
4-(3-fluorophenyl)-N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
1-(furan-2-ylmethyl)-2-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1H-imidazole