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8-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-{[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-phenyl-1,3,4-oxadiazole
2,2-dimethyl-1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(furan-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-6-carboxamide
1-[4-(morpholine-4-carbonyl)piperidin-1-yl]-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
1-(3-phenylpropyl)-4-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-1,4-diazepane
1-(1-cyclobutylpiperidin-3-yl)-4-[3-(trifluoromethyl)phenyl]piperazine
4-[2-(4-fluorophenoxy)ethyl]-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-5-one
N-(2-hydroxypropyl)-2-(4-methoxyphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
5-{[3-(hydroxymethyl)piperidin-1-yl]methyl}-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
6-oxo-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-(3-fluorophenyl)-6,6-dimethyl-N-[(6-methylpyridin-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-methyl-3-[(5-methyl-1,2-oxazol-3-yl)methyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-methyl-6-propyl-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]pyrimidin-4-amine
8-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1-(2-methoxyethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(1H-indazol-1-yl)propyl]-3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
3-hydroxy-1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
2-[methyl({4-methyl-5-[1-(2-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
(1S,5R)-3-[2-(morpholin-4-yl)-2-oxoethyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
8-chloro-3-[2-(1-methylpiperidin-2-yl)ethyl]-3,4-dihydroquinazolin-4-one
{3-ethyl-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}methanol
1-(2-fluoro-6-methoxybenzoyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
4-(dimethylamino)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]butanamide
2-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyrazine
[(3R,4S)-1-[(3-fluoro-2-methylphenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
2-hydroxy-3-methoxy-N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)benzamide
5-[1-(2-ethylbutyl)-4-hydroxypiperidin-4-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-benzofuran-2-carboxamide
4-(1-hydroxyethyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
(3R,4R)-3-cyclopropyl-4-methyl-1-(5-methylthiophene-3-carbonyl)pyrrolidin-3-ol
N-[2-(1,3-benzothiazol-2-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(naphthalen-2-yloxy)acetamide
[1-(5-{[(5-methylfuran-2-yl)methyl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
methyl[2-(piperidin-1-yl)ethyl][(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(2-fluoroethyl)-5-methoxybenzamide
3-cyclopropyl-1-(2-methoxyphenyl)-3-(1,3-thiazol-2-ylmethyl)urea
2-cyclopropyl-N-[cyclopropyl(4-methoxyphenyl)methyl]pyrimidine-5-carboxamide
1-[(2-methoxyphenyl)methyl]-N3-(3-methylbutyl)-4-oxo-N5-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-[(4-methoxyphenyl)methyl]-N-[2-(pyridin-3-yloxy)propyl]-1,2-oxazole-5-carboxamide
N-(1-{7-[(3-ethoxy-4-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)furan-2-carboxamide
2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
5-benzyl-4-(3-hydroxypropyl)-1-(2-methylphenyl)piperazin-2-one
5-benzyl-4-(1H-imidazol-4-ylmethyl)-1-(3-methoxyphenyl)piperazin-2-one
3-({2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-4,6-dimethyl-1,2-dihydropyridin-2-one
2-({4-[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)-5-methylpyrazine
ethyl 2-({8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}amino)benzoate