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N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-5-[(dimethylamino)methyl]-N-methyl-1,3,4-oxadiazole-2-carboxamide
4-{3-[2-(pentan-2-yl)-1H-imidazol-1-yl]propyl}morpholine
2-(methylsulfanyl)-5-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyrimidine
5-(methoxymethyl)-N-[3-(methylsulfanyl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[1-(1H-pyrazol-1-yl)propan-2-yl]pyridin-2-amine
N-methyl-3-propyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-5-carboxamide
2-{[(5-ethylpyridin-2-yl)methyl](methyl)amino}acetic acid
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-2-methylpyridine-3-carboxamide
8-(2,6-dimethoxypyrimidine-4-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decane
4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-N-[1-(3-propyl-1,2,4-oxadiazol-5-yl)ethyl]benzamide
3-{1-[(1-methanesulfonylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}pentan-3-amine
5-(4-chlorophenyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2,4-triazin-3-amine
3-[1-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]pyridine
N-benzyl-N-methyl-3-{1-[2-(morpholin-4-yl)propanoyl]piperidin-4-yl}propanamide
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(ethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
5-fluoro-3-methyl-2-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}-1H-indole
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-(2-phenylethyl)propanamide
1-(2,3-dihydro-1H-inden-2-yl)-5-[2-(ethylsulfanyl)ethyl]-1H-1,2,4-triazole
4-[1-benzyl-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1-methylpiperidin-4-ol
1-cyclohexyl-4-[(2-methoxyethyl)carbamoyl]-1,4-diazepane-6-carboxylic acid
4-{[1-(furan-3-carbonyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
1-{4-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]piperidin-1-yl}ethan-1-one
N-(2-methylpropyl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
2-[methyl(1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)amino]ethan-1-ol
N-(5-{2-cyano-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}-2-methylphenyl)cyclopropanecarboxamide
3-({1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]pyrrolidin-3-yl}methyl)benzamide
1-cyclopentyl-3-(2-fluorophenyl)-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]pyrrolidine-2,5-dione
5-[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]-4-phenyl-1-(pyrrolidin-3-yl)-1H-imidazole
methyl 4-{[2-(2-acetamidoethyl)piperidin-1-yl]methyl}-5-methyl-1,2-oxazole-3-carboxylate
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
3-({[(1-benzyl-1H-pyrazol-4-yl)methyl]amino}methyl)-6-chloro-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
2-[(3-chlorophenyl)methyl]-4-{4-[(2,4-difluorophenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-(3,5-dimethyl-4-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}-1H-pyrrol-2-yl)ethan-1-one
N-[(3R,4S)-1-cyclopentyl-4-(propan-2-yl)pyrrolidin-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
4-pentanamido-N-[3-(pyridin-3-yloxy)propyl]benzamide
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-[(3,4-difluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
(3S,7S,8aS)-7-{[(4-tert-butylphenyl)methyl]amino}-3-[(4-chlorophenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-(2-ethyl-1H-imidazol-1-yl)-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-{1-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidin-3-yl}acetamide
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)amine
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-(quinolin-4-ylmethyl)pyrrolidine-2-carboxamide
6-(4-fluoro-2-methoxyphenyl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
2-amino-8-[4-(ethylamino)pyrimidin-2-yl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
5-[(4,6-dimethyl-1-benzofuran-3-yl)methyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-(2-methoxyethyl)-1-{1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
8-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
5-(3-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}phenoxy)-1-azabicyclo[3.2.1]octane
4-(3-hydroxy-3-methylbutyl)-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)benzamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-(cyclopropylmethyl)-5-(2-methylpent-4-en-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole