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1-(oxan-3-yl)-5,5-diphenylpiperidin-2-one
2-cyclopropyl-8-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl 2-{1-[(4-{[(3,4-dimethoxyphenyl)methyl](methyl)amino}quinazolin-2-yl)methyl]-3-oxopiperazin-2-yl}acetate
(3aR,6aR)-2-[(3-chlorophenyl)methanesulfonyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,7S,8aS)-7-{[(2,5-dimethylphenyl)methyl]amino}-3-[(1R)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-(2,4-difluorophenyl)-3-{[ethyl(oxan-4-yl)amino]methyl}benzamide
3,5-dimethyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
6-{[3-(piperidin-1-yl)pyrrolidin-1-yl]methyl}naphthalen-2-ol
(3S,9aR)-3-(4-aminobutyl)-8-[(3-methylphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
4-{1-[4-(benzyloxy)butanoyl]piperidin-3-yl}benzoic acid
2-methoxy-N-[1-(4-methylphenyl)-5-oxopyrrolidin-3-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-{[(3R,4R)-4-(azepan-1-yl)-3-hydroxypiperidin-1-yl]methyl}-6-methyl-4H-chromen-4-one
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}propanamide
1-{5-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
5-{1-[3-(2-methyl-1H-imidazol-1-yl)propyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
(4aS,7aR)-1-(6-aminopyridine-3-carbonyl)-4-cyclobutanecarbonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-1λ6-thiomorpholine-1,1-dione
4-tert-butyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
2-ethoxy-3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N,5-dimethyl-1-[(methylcarbamoyl)methyl]-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
N-ethyl-N-methyl-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-[2-(1,3-thiazol-2-yl)ethyl]acetamide
1,7-dimethyl-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-indole-2-carboxamide
(2R,3R)-3-amino-1'-(3-methyl-1H-pyrazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(methoxymethyl)-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}cyclobutane-1-carboxamide
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-2,3,6-trimethylquinoline-4-carboxamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
N-benzyl-5-[(3-methoxypropyl)amino]-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-[2-(3-fluorophenyl)ethyl]-2-[4-(4-{[(5-methylfuran-2-yl)methyl]amino}piperidin-1-yl)phenyl]acetamide
N,N,4-trimethyl-5-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]pyrimidin-2-amine
N-{[(2S,4S)-4-fluoro-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl]methyl}pyrrolidine-1-carboxamide
3-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-(5,7,8-trimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
ethyl({[2-(prop-2-en-1-yloxy)phenyl]methyl})(pyridin-2-ylmethyl)amine
3-acetyl-N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1H-pyrazole-5-carboxamide
1-{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
3-methanesulfonyl-N-[(3R,4S)-1-(2-methoxyethyl)-4-phenylpyrrolidin-3-yl]propanamide
1-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}-2-phenylethan-1-ol
1-tert-butyl-N-(1-cyclohexyl-1H-pyrazol-5-yl)-5-oxopyrrolidine-3-carboxamide
4-(2-methylphenoxy)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-3-carbonitrile
3-methyl-6-{5-[2-(trimethyl-1H-pyrazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
N-(oxolan-2-ylmethyl)-3-(1H-pyrazol-1-ylmethyl)-N-(pyridin-2-ylmethyl)benzamide
2-methoxy-5-[(3-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidin-1-yl)methyl]phenol
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-4-(morpholine-4-sulfonyl)phenol
N-[1-(pyrazin-2-yl)piperidin-4-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
3-(2-methoxyphenyl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
[(4-fluorophenyl)methyl]({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amine
2-({2-amino-6-[(1R,5S)-3,8-diazabicyclo[3.2.1]octan-3-yl]pyrimidin-4-yl}amino)ethan-1-ol