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N-{[2-(diethylamino)pyridin-3-yl]methyl}-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
2-methyl-4-(5-{1-[(2S)-oxolan-2-ylmethyl]-4-phenyl-1H-imidazol-5-yl}thiophen-2-yl)but-3-yn-2-ol
5-cyclopropanecarbonyl-1'-(3-phenyl-1,2,4-oxadiazol-5-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
1-{[1-(2-methoxyphenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}azepane
N-cyclopropyl-1-phenyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
1-[(2S,4S)-4-amino-1-methylpyrrolidine-2-carbonyl]-4-phenylpiperidine-4-carbonitrile
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}({[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl})methylamine
8-(5-fluoro-2-methoxybenzoyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[(1-cyclooctylpyrrolidin-3-yl)methyl]-2-methanesulfonamidoacetamide
2-[4-(2H-1,3-benzodioxol-5-yl)-3-butyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-cyclobutylacetamide
6-ethyl-N,N-dimethyl-2-[2-(pyridin-3-yl)pyrimidin-5-yl]quinoline-4-carboxamide
2-(4-chlorophenyl)-5-[(4-fluorophenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
[(4-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-2-yl}phenyl)methyl]dimethylamine
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(1H-pyrazol-1-yl)propan-1-one
propyl 3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxylate
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-{[(2R)-2-hydroxypropyl]sulfamoyl}benzamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-6-methoxy-3,4-dihydroquinazolin-4-one
3-tert-butyl-4-{6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4,5-dimethyl-6-[4-(pyridin-4-yl)piperazin-1-yl]pyrimidin-2-amine
2-{[3-(2-methylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}ethan-1-one
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[3-(pyridin-4-yl)propyl]pyridin-2-amine
3-[(5,6-dichloro-1H-1,3-benzodiazol-2-yl)methyl]-2,3-dihydro-1,3-benzoxazol-2-one
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]({[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl})amine
[2-ethoxy-5-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenyl]methanol
3-(2-phenoxyethyl)-8-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}thiomorpholine
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-1,4-diazepan-5-one
4-[(3-methylphenyl)methyl]-1-(thiophen-3-ylmethyl)-1,4-diazepan-5-one
8-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
6-({1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]hex-5-en-2-yl}oxy)pyridine-2-carbonitrile
(2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-thiazol-4-yl)methanol
N-[(3R,4S)-1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-4-cyclopropylpyrrolidin-3-yl]-2-(dimethylamino)acetamide
9-(1-ethyl-1H-pyrazole-3-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(5-fluoro-2-methoxyphenyl)-2-methylquinazoline
1-[3-(4,5-dihydro-1H-imidazol-2-yl)phenyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
(1R,5R)-6-[2-(4-fluorophenoxy)ethyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N'-(2,4-dimethylphenyl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]propanediamide
5-[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-4-methyl-1,2,3-thiadiazole
ethyl 2-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]-1,3-oxazole-4-carboxylate
(3S,4R)-1-(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
N-{[2-(diethylamino)pyridin-3-yl]methyl}-5-methylpyrazine-2-carboxamide
(1R,2R,6S,7S)-N-{2-[2-(pyridin-2-yl)ethyl]phenyl}-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
methyl[(5-methylfuran-2-yl)methyl]{[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
4,5-dimethyl-2-[5-(pyrazine-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1H-1,3-benzodiazole
1-[(2-chlorophenyl)methyl]-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1H-1,2,3-triazole-4-carboxamide
6-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}pyridine-2-carboxylic acid
4-hydroxy-N-(2-hydroxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide