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4-(3-aminopropanoyl)-5-benzyl-1-(4-methylphenyl)piperazin-2-one
(3S,4R)-N,N-dimethyl-1-(1-methyl-4-phenylpiperidine-4-carbonyl)-4-(propan-2-yl)pyrrolidin-3-amine
(3R,4R)-3-cyclobutyl-4-methyl-1-(trimethyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-ol
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2,7,8-trimethylquinoline-4-carboxamide
(2S)-2-(methoxymethyl)-N-{4-[2-(pyridin-2-yl)ethyl]phenyl}pyrrolidine-1-carboxamide
2-{1-[(5-methylfuran-2-yl)methyl]-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperazin-2-yl}ethan-1-ol
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-ethyl-1,2-oxazole-4-carboxamide
1-[7-(6,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
3-chloro-4-{[1-(cyclohexylmethyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
N-ethyl-2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-(propan-2-yl)-1,3-oxazole-4-carboxamide
5-[3-({[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino}methyl)pyrrolidin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
5-[3-(4-fluorophenoxy)azetidine-1-carbonyl]-1-methyl-3-propyl-1H-pyrazole
(3S,4R)-1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)-4-(propan-2-yl)-1,2,3-thiadiazole-5-carboxamide
2-(piperazin-1-yl)-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}acetamide
3-{1-[4-(methylamino)pyrimidin-2-yl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(3-methoxypropyl)-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}propanamide
N-{[1-(3,5-dimethylphenyl)cyclopentyl]methyl}-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
1-(cyclohexylmethyl)-N5-(2,2-diphenylethyl)-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
dimethyl(2-{2-[1-(4-methylquinolin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
N-[(3S,4R)-4-(propan-2-yl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-3-yl]methanesulfonamide
3-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]-3,9-diazaspiro[5.6]dodecan-10-one
3-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)propanamide
5-{4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1-methyl-1H-pyrrol-3-amine
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-4-(piperidin-1-yl)butanamide
1-{2-[3-(furan-2-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]ethyl}azepan-2-one
5-{[2-(4-methanesulfonylphenyl)-1H-imidazol-1-yl]methyl}-2,1,3-benzothiadiazole
1-(2-methylphenyl)-4-(6-oxo-1,6-dihydropyridine-3-carbonyl)piperazin-2-one
3-[(1-benzoylpiperidin-4-yl)amino]-2,3-dihydro-1λ6-thiophene-1,1-dione
3-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]quinoline
2-{[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}pyridine
1-{2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-2-oxoethyl}-3,3-dimethylurea
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}acetamide
4-fluoro-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzene-1-sulfonamide
2-[(cyclopropylmethyl)sulfanyl]-1-{4-[(2-methylphenyl)methyl]piperazin-1-yl}ethan-1-one
2-(5-{6-amino-5-cyano-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridin-2-yl}thiophen-3-yl)acetic acid
1-(3-chlorophenyl)-5-methyl-4-(quinolin-5-ylmethyl)piperazin-2-one
2-[2,6-dimethyl-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
(2-{2-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
methyl (2S,4R)-4-(3-chloro-5-methoxybenzamido)-1-methylpyrrolidine-2-carboxylate
1-ethyl-3-methyl-8-[(1-methyl-1H-indol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-2-{8-methyl-3-oxo-2,8-diazaspiro[4.5]decan-2-yl}-N-[2-(phenylsulfanyl)ethyl]acetamide
1-[(5-ethylpyridin-2-yl)methyl]-4-(2-methylquinolin-6-yl)piperidin-4-ol
5-acetyl-N-ethyl-N-[(2-fluorophenyl)methyl]thiophene-3-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-fluoro-4-methoxy-N-(pyridin-3-ylmethyl)benzamide
N-{2-[(4-fluorophenyl)formamido]ethyl}oxane-2-carboxamide
N-{2-[3-cyclopropyl-1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-N-methylmethanesulfonamide
2,4-difluoro-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzene-1-sulfonamide
methyl 3-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-oxopropanoate