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1-(2-chlorophenyl)-3-{1-[1-(3-methylpentanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
3-(1-benzofuran-2-ylmethyl)-5-(piperidin-4-yl)-5-propylimidazolidine-2,4-dione
2-[3-cyclopentyl-5-(2-phenoxyethyl)-1H-1,2,4-triazol-1-yl]acetic acid
4-cyano-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)oxane-4-carboxamide
(2S)-2-{[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}-3-phenylpropan-1-ol
4-[2-(3-chlorophenyl)-2-hydroxyacetyl]-1-(3-methoxyphenyl)piperazin-2-one
N-cyclohexyl-N-methyl-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
5-methyl-4-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-1-(2-methylphenyl)piperazin-2-one
N-[1-(3-methoxyphenyl)ethyl]-N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
(3-{2-[1-(3-fluoro-4-methylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
2-methoxy-N-({5-methyl-2-[3-(oxane-4-amido)phenyl]-1,3-oxazol-4-yl}methyl)pyridine-3-carboxamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[(4-fluorophenyl)methyl]-N-methylacetamide
5-(3-ethyl-1,2,4-oxadiazol-5-yl)-2-(pyridin-4-yl)pyrimidine
N-{2-[(1,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)formamido]ethyl}acetamide
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-6-carboxamide
N-[2-(3-chlorophenyl)ethyl]-5-(4-methylpiperidine-1-carbonyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethan-1-one
7-(1,3-benzothiazol-2-yl)-4-(pyrazine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2,3-dimethyl-7-{[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-indole
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
3-{3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl}propanamide
3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-6-(4-methylpiperazin-1-yl)pyridazine
N-[1-(1-cyclopentanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-2-methoxy-2-phenylacetamide
4-{1-[2-(azocan-1-yl)acetyl]piperidin-3-yl}benzoic acid
1-[3-(2-fluorophenyl)pyrrolidin-1-yl]-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propan-1-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[1-(1H-imidazol-1-ylmethyl)cyclopropanecarbonyl]piperidin-3-ol
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2,3-dihydro-1H-indene-1-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-3-(3-hydroxy-3-methylbutyl)benzamide
3-[4-(4-methoxy-2-methylphenyl)-1H-pyrazol-1-yl]propanamide
4-methyl-1-(6-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)piperidine-4-carbonitrile
(2,1,3-benzoxadiazol-5-ylmethyl)[4-(2-methyl-1H-imidazol-1-yl)butan-2-yl]amine
dimethyl(2-{2-[1-(pyrimidin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
3-{4-[(2-chloro-4-ethoxy-5-methoxyphenyl)methyl]piperazin-1-yl}-6-methylpyridazine
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
N1-ethyl-N2-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-1,2-dicarboxamide
[(5-chloro-3-methyl-1H-indol-2-yl)methyl](1,4-dioxan-2-ylmethyl)methylamine
2-{1-[(4-fluorophenyl)methyl]-4-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
5-fluoro-4-(pyrrolidin-1-yl)-2-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidine
4-(1-benzothiophen-2-ylmethyl)-11-[(3-hydroxy-2,2-dimethylpropyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-{[1-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)pyrrolidin-3-yl]methyl}benzamide
{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
7-chloro-2-{[6-(hydroxymethyl)-1,4-oxazepan-4-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
5-(4-fluorophenyl)-3-(3-methoxypiperidin-1-yl)-1,2,4-triazine
(3S,4S)-3-({[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}(methyl)amino)-4-hydroxy-1λ6-thiolane-1,1-dione
3-{1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}-N-[(2-fluorophenyl)methyl]propanamide
4-ethyl-3-({1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2-methylphenol
4-{3-[2-(methoxymethyl)piperidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
(3aR,6aS)-5-(3-cyano-5-fluorobenzoyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[(2S)-1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol