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1-{4-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]phenyl}ethan-1-one
3-cyano-5-fluoro-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylbenzamide
2-{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]pyrrolidin-2-yl}-1,3-thiazole
3-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-sulfonyl]-N-(2-ethoxyethyl)benzamide
4-phenyl-N-{[1-(pyridine-3-carbonyl)piperidin-3-yl]methyl}benzamide
N-{[4-(morpholin-4-yl)phenyl]methyl}-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)acetamide
4-(1-{[3-fluoro-4-(trifluoromethyl)phenyl]methyl}azetidin-3-yl)pyridine
2-[(4-methylphenyl)amino]-2-phenyl-N-(pyridin-4-ylmethyl)propanamide
2-(1H-1,2,3-benzotriazol-1-yl)-N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)acetamide
2-methyl-1-{2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}-1,4-diazepan-5-one
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
3-(dimethylsulfamoyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-5-[(3-phenylpropyl)amino]benzamide
3-[(2-methoxyphenyl)methyl]-1-methyl-5-(3,3,3-trifluoropropyl)-1H-1,2,4-triazole
2-(dimethylamino)-N-(2-methanesulfonamidoethyl)-2-(3-methylphenyl)acetamide
3-(6-methoxypyridin-2-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
2-ethyl-8-(2-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(2-propoxyethyl)-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]-2-(morpholin-2-yl)acetamide
4-{[2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperazine-2-carboxylic acid
S-[2-(2-ethoxyacetyl)-1,2,3,4-tetrahydroisoquinolin-6-yl]-3-hydroxybutane-1-sulfonamido
N,N-dimethyl-5-{[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyridin-2-amine
2-(6-oxo-1,6-dihydropyridine-3-carbonyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(4-methyl-1H-imidazol-2-yl)ethyl]amine
2-(but-3-enoyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
methyl 4-{7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}benzoate
3-(3-methoxybenzoyl)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)-4-({[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)pyrrolidine-2-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5,6-dimethylpyrimidin-4-amine
N-(2-{7-[(3-ethoxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
2-(2-hydroxyethyl)-8-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
2-{1-cyclopentyl-4-[1-(2-phenylethyl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
5-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}-N-phenylpyrimidin-2-amine
6-(2-chlorophenyl)-N,N-dimethyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(8R,9aS)-8-hydroxy-2-[2-(3-methoxyphenyl)ethyl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
1-cyclobutanecarbonyl-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxamide
6-{[4-(pentan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-1H-indole
2-butanoyl-7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-6-one
3-hydroxy-1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
(4aS,7aR)-1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2-hydroxyphenyl)-1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}propan-1-one
(3S,4S)-4-(2,3-dihydro-1H-isoindol-2-yl)-1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}pyrrolidin-3-ol
N,N-dimethyl-5-[3-(4-methylpiperidine-1-carbonyl)phenyl]thiophene-2-carboxamide
4-(4-benzyl-1H-pyrazol-5-yl)-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidine
7-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[(2-fluorophenyl)methyl]-1-methyl-5-{[3-(morpholin-4-yl)propyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-(cyclopropylmethyl)-2-[2-(3-methylphenoxy)acetyl]-2,7-diazaspiro[4.5]decan-6-one
{[(3S,4R)-1-(3,6-dimethylpyrazin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-(prop-2-en-1-yl)-1H-1,3-benzodiazole-5-carboxamide
2-[4-(hydroxymethyl)phenyl]-1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethan-1-one