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methyl 4-(4-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
methyl 2-chloro-5-({[3-(2-oxopyrrolidin-1-yl)propyl]carbamoyl}amino)benzoate
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
{1-[(3,4-dichlorophenyl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
4-[2-(4-oxo-3,4-dihydroquinazolin-3-yl)ethyl]benzene-1-sulfonamide
N,1-dimethyl-N-(thiophen-3-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
N-cyclopentyl-2-{[2-(2,3-dihydro-1H-indol-1-yl)ethyl]amino}propanamide
[4-({3-propyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}sulfonyl)phenyl]urea
4-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
1-[3-(3-{[4-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)propyl]piperidine
11-(benzylamino)-4-[(2-methoxynaphthalen-1-yl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-1-methylpiperidine-4-carboxamide
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-4,4,4-trifluorobutan-1-one
4-ethyl-5-methyl-2-[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]pyrimidine
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(4-fluorobenzoyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-[4-(1,3-benzoxazol-2-yl)piperazine-1-carbonyl]pyrazin-2-ol
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}acetamide
3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{[1-(propan-2-yl)piperidin-4-yl]methyl}piperazine
2-(5-acetylthiophen-3-yl)-N-cyclohexyl-N-(pyridin-2-ylmethyl)acetamide
2-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]acetic acid
11-(isoquinolin-5-ylmethyl)-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
2-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N,7-bis(cyclopropylmethyl)-8-oxo-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-4-(1H-1,2,4-triazol-1-yl)butanamide
2,4-dimethyl-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}pyrimidine-5-carboxamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-N-(2-methoxyethyl)propanamide
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(2-methanesulfonylethyl)piperazin-1-yl]ethan-1-one
methyl (2S)-1-[7-(3-methoxypropanamido)-1-methyl-2-phenyl-1H-1,3-benzodiazole-5-carbonyl]pyrrolidine-2-carboxylate
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-3-[(dimethylamino)methyl]benzamide
3-methoxy-5-{1-oxa-8-azaspiro[4.6]undecane-8-carbonyl}benzoic acid
3-{ethyl[(2-hydroxy-6-methoxyquinolin-3-yl)methyl]amino}-1λ6-thiolane-1,1-dione
1-[3-(1H-imidazol-2-yl)benzoyl]-4-methanesulfonyl-1,4-diazepane
1-ethyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-5-oxopyrrolidine-3-carboxamide
3-(4-hydroxyphenyl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}pyrazin-2-amine
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-[2-(pyridin-2-yl)ethyl]acetamide
N-[(2S,4R,6S)-2-benzyl-6-(4-hydroxy-3,5-dimethoxyphenyl)oxan-4-yl]acetamide
2-(prop-2-en-1-yl)-9-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-benzoyl-6-methyl-5-[5-(1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
3-[(2,2-diethylmorpholin-4-yl)methyl]-6-methoxy-1,2-dihydroquinolin-2-one
N-[1-(4-hydroxyphenyl)propyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
1-(1,3-benzoxazol-2-yl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
ethyl[(4-methoxyphenyl)methyl]{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
5-(2-butyl-4-methyl-3-oxopiperazine-1-carbonyl)-2,3-dimethylbenzene-1-sulfonamide
2-(morpholin-4-yl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]benzamide
5-{[benzyl(methyl)amino]methyl}-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
8-{5-amino-[1,2,4]triazolo[4,3-c]pyrimidin-7-yl}-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one