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(1S,5R)-6-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[4-(dimethylamino)oxan-4-yl]methyl}-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-ethyl-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
[1-(1H-indol-3-ylmethyl)-4-[(4-methoxyphenyl)methyl]piperidin-4-yl]methanol
2-[5-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-1-yl]pyridine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-4-(pyridin-4-yl)pyrimidin-2-amine
3-({4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenol
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2-(thiophen-2-yl)pyrimidine-5-carboxamide
1-[(4-fluorophenyl)methyl]-4-[3-(1-methylpiperidin-2-yl)propanoyl]piperazin-2-one
9-[2-(propylsulfanyl)acetyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[4-(1H-pyrazol-1-yl)butan-2-yl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
6-{[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-benzyl-N-ethyl-5-[(2-methoxyethyl)(methyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[3-(5-chloro-1H-1,3-benzodiazol-2-yl)propyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
5-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-4-yl}-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
N-[(3-hydroxypyrrolidin-3-yl)methyl]-5-(4-methoxyphenyl)furan-2-carboxamide
5-(4-chloro-2-methoxyphenoxymethyl)-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-1-(2-methylpropyl)piperidin-4-amine
methyl (1R,3S,3aR,6aS)-1-(2-methoxy-2-oxoethyl)-5-methyl-4,6-dioxo-3-(thiophen-2-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
(2S)-1-{3-[(2-methylprop-2-en-1-yl)oxy]benzoyl}pyrrolidine-2-carboxamide
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-tert-butyl-1-methyl-1H-pyrazole-5-carboxamide
3,5-difluoro-2-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyridine
N-{2-[(1-cyclopentyl-6-oxopiperidin-3-yl)formamido]ethyl}-4-fluorobenzamide
4-methoxy-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)benzamide
4-[5-({[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
3-(methylsulfanyl)-1-[2-(2-phenylethyl)morpholin-4-yl]propan-1-one
1-(2-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}ethyl)pyrrolidin-2-one
1-[(2R)-2,3-dihydroxypropyl]-2-oxo-3-(pentan-3-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
1-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-3-(furan-2-ylmethyl)urea
N-[2-(1H-imidazol-4-yl)ethyl]-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
(4S)-3-(2-oxo-2-{1,5,7-trimethyl-3,7-diazabicyclo[3.3.1]nonan-3-yl}ethyl)-4-(propan-2-yl)-1,3-oxazolidin-2-one
2-(9-methyl-9H-carbazol-3-yl)-N-[2-(6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]acetamide
N-(cyclopropylmethyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
2-cyclopropyl-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]quinoline-4-carboxamide
(2S)-2-[4-(2-phenylethyl)piperazine-1-carbonyl]pyrrolidine-1-carboxamide
2-[1-(2,2-dimethylpropyl)-4-[(3-methyl-1H-pyrazol-5-yl)methyl]piperazin-2-yl]ethan-1-ol
2-[2-(1H-imidazol-1-yl)ethyl]-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine
4-{7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}benzene-1-sulfonamide
N-ethyl-3,4,7-trimethyl-N-(oxan-2-ylmethyl)-1H-indole-2-carboxamide
methyl 2-{4-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-2-oxopiperazin-1-yl}acetate
5,6-dimethyl-2-[3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carbonitrile
5-cyclobutyl-N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,3,4-oxadiazol-2-amine
3-(2,4-dimethoxybenzoyl)-1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidine
N-(1,4-dioxan-2-ylmethyl)-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-(2-chlorophenyl)-3-[1-(1-propanoylpiperidin-4-yl)-1H-pyrazol-5-yl]urea
1-(5-ethyl-1,3,4-oxadiazol-2-yl)-3-propoxypiperidine
2-cyclohexyl-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1,3-benzoxazole-6-carboxamide
1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
4-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide