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N-(3-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)acetamide
N-[(2-ethoxyphenyl)methyl]-N,1-diethyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[1-(3-methylbutyl)-4-(pyridin-2-ylmethyl)piperazin-2-yl]ethan-1-ol
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(1-methyl-1H-indol-3-yl)acetamide
3-[2-(dimethylamino)ethyl]-5-[1-(1-methylpiperidine-3-carbonyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
4-(2,6,8-trimethylquinoline-4-carbonyl)-1λ6-thiomorpholine-1,1-dione
N-benzyl-N-ethyl-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
(2S,4S,5R)-4-[(1-carboxy-1-methylethyl)carbamoyl]-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
2-amino-6-(4-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)-3,4-dihydropyrimidin-4-one
N-({1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-hydroxyazepan-4-yl}methyl)cyclopropanesulfonamide
3-[2-(2-fluorophenyl)ethyl]-1-(5-propyl-1,2-oxazole-4-carbonyl)piperidine
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-2-(1H-indol-1-yl)ethan-1-one
2-(2-{1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
5-(butan-2-yl)-N-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(2-methoxyphenyl)methyl]-N3-(3-methylbutyl)-4-oxo-N5-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-(piperazin-1-ylmethyl)piperidin-2-one
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(2-oxo-1,2-dihydroquinoxalin-1-yl)acetamide
N-(4-fluoro-2-methylphenyl)-2-[(3-methyl-1H-pyrazol-5-yl)formamido]propanamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
3-[2-(4-fluorophenyl)ethyl]-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
1-[2-(piperidin-1-yl)ethyl]-6-[3-(pyridin-2-yl)propanoyl]-3-(pyridin-4-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-(3-methoxyphenoxymethyl)-N-(2,2,2-trifluoroethyl)-1,3-oxazole-4-carboxamide
7-hydroxy-2-oxo-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-1,2,3,4-tetrahydroquinoline-6-carboxylic acid
(1R,5R)-N,N-dimethyl-6-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
4-(4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}phenyl)-2-methylbutan-2-ol
N-(2-ethyl-2-methyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)-2-methyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
5-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
5,6-dimethyl-3-(pyridin-2-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
3-tert-butyl-1-({1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl}methyl)urea
3-(1H-1,3-benzodiazol-1-yl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
3-(3-hydroxy-3-methylbutyl)-N-[(1-methyl-5-oxopyrrolidin-2-yl)methyl]benzamide
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-(4-methylphenyl)-1H-pyrazole-3-carboxamide
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-1-(propan-2-yl)piperidine-4-carboxamide
1-cyclobutanecarbonyl-N-[(dimethyl-1,3-thiazol-2-yl)methyl]piperidine-4-carboxamide
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
5-(2,4-dimethoxypyrimidin-5-yl)-8-methoxyquinoline
1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}azepan-2-one
1-[(4aR,8aR)-7-[(2-chloro-4-fluorophenyl)methyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
3-methyl-8-[(1-methyl-1H-imidazol-2-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
[1-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-3-propylpiperidin-3-yl]methanol
N-(4-{[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}phenyl)cyclopropanecarboxamide
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-5-ethyl-1,3,4-oxadiazol-2-amine
N-ethyl-6-(4-ethylphenyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[3-({[(4-fluorophenyl)methyl](oxolan-2-ylmethyl)amino}methyl)pyridin-2-yl]-2,2-dimethylpropanamide
N-[(2R,3R)-2-ethoxy-1'-(2-methoxyquinoline-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-(3-methylpyridin-4-yl)-4-[2-(pyrrolidin-3-yl)benzoyl]-1,4-diazepane
(1S,5R)-3-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[2-(5-acetylthiophen-3-yl)acetyl]-1-(3,5-dimethylphenyl)piperazin-2-one