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4-ethyl-1-methyl-3-{1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
ethyl 4-{[2-(2,3-dihydro-1H-indol-1-yl)ethyl]amino}piperidine-1-carboxylate
N-[2-(2-fluorophenyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]ethyl]-N-methylthiophene-3-carboxamide
3,5-dichloro-4-[1-(2,6-dimethoxypyridin-3-yl)-1H-imidazol-2-yl]pyridine
1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
3,3-dimethyl-N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
N-ethyl-4-oxo-1-(2-phenylethyl)-5-(4-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-(thiophen-2-ylmethyl)acetamide
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
[(4-ethylphenyl)methyl](methyl){2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
1-{[5-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-2-methoxyphenyl]methyl}-1H-pyrazole
4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]-1-[(2S)-pyrrolidine-2-carbonyl]piperidine
2-{4-[3-(trifluoromethyl)phenoxymethyl]phenyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
methyl (2S,3S)-2-(3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamido)-3-methylpentanoate
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-[2-(2-methylphenyl)ethyl]piperidine
(3R,4S)-4-{4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1,4-diazepan-1-yl}oxolan-3-ol
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-2-cyclopentylacetamide
(3aS,6aS)-2-{[4-(2-fluorophenyl)phenyl]methyl}-5-(2-hydroxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-(2-fluorophenyl)-3-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]propanamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,3-oxazole-4-carboxamide
2-methyl-8-[(6-phenoxypyridin-3-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3R,4R)-4-methyl-3-(propan-2-yl)-1-(propane-2-sulfonyl)pyrrolidin-3-ol
2-[2-({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
3-{5-[2-(2-methyl-1H-indol-3-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
5-(1-ethyl-1H-indole-5-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-(1-methyl-1H-pyrazole-5-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
8-(2,6-dimethylpyridin-4-yl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
ethyl 1-({7-fluoro-1-[(3-methoxyphenyl)methyl]-2-oxo-1,2-dihydroquinolin-3-yl}methyl)piperidine-4-carboxylate
1-ethyl-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-5-oxopyrrolidine-3-carboxamide
methyl 1-[(3R,5S)-1-[(3-hydroxyphenyl)methyl]-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-2-methoxy-N-(oxolan-2-ylmethyl)benzamide
N-(butan-2-yl)-2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-[(3-methylthiophen-2-yl)methyl]acetamide
4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}morpholine-2-carboxylic acid
(3S,4S)-1-[2-(cyclopentylcarbamoyl)ethyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]-2-(furan-2-yl)ethane-1,2-dione
1-[benzyl(methyl)amino]-3-(4-{[4-(propan-2-yl)piperazin-1-yl]methyl}phenoxy)propan-2-ol
N-(4-methoxy-2-methylphenyl)-3-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}propanamide
3-methoxy-1-{4-[4-(3-propoxypiperidine-1-carbonyl)phenoxy]piperidin-1-yl}propan-1-one
4-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
N-(1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}acetamide
2-(4-chloro-1H-pyrazol-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
2-(1,3-dihydroxypropan-2-yl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
2-{[6-(4-cyclohexylpiperazin-1-yl)pyridazin-3-yl]oxy}-1-(thiomorpholin-4-yl)ethan-1-one
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-cyclopropyl-1-[(4-phenylphenyl)methyl]pyrrolidine-2-carboxamide