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{5-[(4-{1-[(2-methoxyethyl)(pyridin-2-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)methyl]furan-2-yl}methanol
N-{[(2S,4S)-1-[2-(2,3-dimethylphenoxy)acetyl]-4-fluoropyrrolidin-2-yl]methyl}ethane-1-sulfonamide
(3aS,6aS)-1-{2-[2-(3-methoxyphenyl)ethyl]benzoyl}-octahydropyrrolo[2,3-c]pyrrole
3-methoxy-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1,2-dihydropyridin-2-one
3-[2-(methylsulfanyl)ethyl]-5-phenylmethanesulfonyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-methyl-3-[4-(3-methylphenyl)piperazin-1-yl]-N-(thian-4-yl)propanamide
1-{4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
5-(dimethylamino)-2-[2-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-oxoethyl]-2,3-dihydropyridazin-3-one
1-{[({4-[2-hydroxy-3-(morpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)amino]methyl}cyclohexan-1-ol
N-methyl-2-oxo-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1,2-dihydroquinazoline-4-carboxamide
2-(1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-imidazol-2-yl)-1H-1,3-benzodiazole
1-(2-methoxyphenyl)-4-[1-(thiophene-3-sulfonyl)piperidin-3-yl]piperazine
7-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-ylmethyl]-4-methyl-2H-chromen-2-one
1-(dimethylamino)-2-[4-(naphthalen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-2-ol
ethyl 1-(4-chlorobenzenesulfonyl)-4-(cyclopropylmethyl)piperidine-4-carboxylate
N-(2-{[benzyl(1,3-thiazol-2-ylmethyl)amino]methyl}quinolin-6-yl)acetamide
1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}hexan-1-one
2-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]-2-azaspiro[4.4]nonane
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-(3-methyl-3-phenylpiperidin-1-yl)propan-1-one
N-(1-{7-[(2-hydroxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-3,5-dimethylbenzamide
(3R,4S)-4-cyclopropyl-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]pyrrolidin-3-amine
1-[(3-methoxyphenyl)methyl]-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-(adamantan-1-ylsulfanyl)-1-[3-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
(1S,5R)-3-(pyridin-4-ylmethyl)-6-{[2-(trifluoromethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)furan-2-carboxamide
6-[4-(azepan-1-yl)butyl]-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
3-({1-[(2,6-difluorophenyl)methyl]piperidin-4-yl}methyl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(4-ethoxyphenyl)methyl]-4-(3-propyl-1H-pyrazole-5-carbonyl)piperazine
(5-{[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}furan-2-yl)methanol
4-{[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}benzoic acid
N-[5-(ethylsulfanyl)-1,3,4-thiadiazol-2-yl]-2-[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidin-1-yl]acetamide
2-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-3-yl}benzoic acid
2-cyclopropanecarbonyl-8-(2-hydroxypyridine-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(2S,6S)-4-methyl-1-[3-(2-phenylethyl)-1,2-oxazole-5-carbonyl]-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
3-{3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-1,2-benzoxazole
2-(4-acetyl-1,4-diazepan-1-yl)-2-(2,4-dimethylphenyl)acetic acid
N4-[2-(4-chlorophenoxy)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
3-cyclopentaneamido-N-[4-(pyrrolidin-1-yl)butyl]benzamide
(1R,4R)-2-{3-[4-(2-methylphenyl)piperazin-1-yl]propyl}-2-azabicyclo[2.2.1]heptane
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,2,7-trimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
3-[(2R,3R,6R)-5-(1H-indole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
(2R)-1-{[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}pyrrolidine-2-carboxamide
2-methyl-6-[2-(pyrrolidin-1-yl)ethyl]-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
1-[4-(furan-3-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]-3-(pyridin-4-yl)propan-1-one
3-{1-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-3-ol
3-(1-propyl-1H-1,2,3-triazol-4-yl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}urea
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}bis(pyridin-3-ylmethyl)amine
5-methyl-2-(1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
2-{[2-(1H-indol-3-yl)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide