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N-(1-cycloheptylpiperidin-3-yl)-3-(4-methyl-1,3-thiazol-5-yl)propanamide
4-(1-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperidin-4-yl)pyridine
1-[1-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperidin-4-yl]piperidin-3-ol
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3aR,6aR)-2-(pyridin-3-ylmethyl)-5-(quinolin-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)urea
1-(3-fluoro-2-methoxybenzoyl)-3-[2-(2-fluorophenyl)ethyl]piperidine
(1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}-4-(2-phenoxyethyl)piperidin-4-yl)methanol
(3S,4R)-1-[(4-methylpiperidin-1-yl)sulfonyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]acetic acid
8-chloro-2-({[3-(pyridin-4-yl)propyl]amino}methyl)quinolin-4-ol
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)furan-3-carboxamide
3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-7-methyl-1H-indole
5-(3-chlorothiophene-2-carbonyl)-N-cyclopropyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[(1-cyclobutanecarbonylpiperidin-4-yl)formamido]-2-(3-hydroxyphenyl)acetic acid
(3R,4S)-4-propyl-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidin-3-amine
3-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydroquinolin-2-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(2-propoxybenzoyl)pyrrolidin-3-yl]methanol
[(2-chlorophenyl)methyl](ethyl)[(2S)-pyrrolidin-2-ylmethyl]amine
3-[3-(2-chlorophenoxymethyl)-4H-1,2,4-triazol-4-yl]pyridine
2-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
7-(3,6-dimethylpyrazin-2-yl)-9-methoxy-4-(oxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{[2-(3,4-dimethoxyphenyl)-7-methylquinolin-3-yl]methyl}piperidine-3-carbonitrile
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl]amine
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]acetamide
methyl 3-{[2-(5-phenyl-4H-1,2,4-triazol-3-yl)acetamido]methyl}-5-[(2E)-3-phenylprop-2-enamido]benzoate
(1S,6R)-3-methyl-9-(1-phenyl-1H-1,2,3-triazole-5-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
2-{5-cyclobutyl-3-[(2,6-dichlorophenyl)methyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-[2-methoxy-5-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
(3R,4S)-4-cyclopropyl-1-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidin-3-amine
5-{6-oxa-9-azaspiro[4.5]decan-9-yl}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-(2-aminopyrimidin-5-yl)-N,N,5,7-tetramethylquinoline-4-carboxamide
3-(1,3-dimethyl-1H-pyrazol-4-yl)-1-[2-(2-methoxyphenyl)ethyl]urea
2-(2-methoxyethoxy)-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
2-[({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]-4,6-dimethylpyridine-3-carbonitrile
2-[3-(aminomethyl)pyrrolidine-1-carbonyl]-N-methyl-N-(2-phenylethyl)-2,3-dihydro-1H-inden-2-amine
N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
8-[3-(3-methoxyphenoxy)propyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
6-[(2,4-dimethoxyphenyl)methyl]-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
6-(3-fluoro-4-methoxyphenyl)-N-(furan-2-ylmethyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(1,3-thiazol-4-yl)ethyl]pyridin-2-amine
(4aS,7aR)-1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-(4-methoxyphenoxy)-N-[2-(pyridin-2-yl)ethyl]benzamide
N-[2-(1H-indol-3-yl)ethyl]-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-amine
1-{2-[4-(2-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydroquinolin-2-one
N-(cyclopropylmethyl)-1-(6-fluoro-4-methylquinazolin-2-yl)azepan-4-amine
1-(morpholin-4-yl)-3-[5-(pyridin-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propan-1-one
N-(2-{7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
(3R)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide